SCHEMBL13633878

SCHEMBL13633878

Cc1ccc2cccnc2c1NS(=O)(=O)c1cc(Cl)c(Cl)s1

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC40A1 Q9NP59 12/20 0.59
MEN1 O00255 4/20 0.50
KMT2A Q03164 4/20 0.50
NFKBIA P25963 2/20 0.47
RELA Q04206 2/20 0.47
TDP1 Q9NUW8 3/20 0.46
ATM Q13315 1/20 0.45
PTGES2 Q9H7Z7 1/20 0.44
THRB P10828 1/20 0.43
BLM P54132 1/20 0.43
CCR4 P51679 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13633842 0.83 NFKBIA (0.68) SLC40A1MEN1KMT2ANFKBIARELA
SCHEMBL13485925 0.82 NFKBIA (0.70) SLC40A1MEN1KMT2ANFKBIARELA
SCHEMBL13633844 0.81 SLC40A1 (0.59) SLC40A1MEN1KMT2ANFKBIARELA
SCHEMBL13633824 0.79 SLC40A1 (0.68) SLC40A1MEN1KMT2ANFKBIARELA
SCHEMBL13633768 0.78 SLC40A1 (0.61) SLC40A1MEN1KMT2ANFKBIARELA
SCHEMBL2055429 0.78 SLC40A1 (0.72) SLC40A1MEN1KMT2ATDP1
SCHEMBL13633855 0.78 NFKBIA (0.67) SLC40A1MEN1KMT2ANFKBIARELA
SCHEMBL13633916 0.76 SLC40A1 (0.72) SLC40A1MEN1KMT2ANFKBIARELA
SCHEMBL13633857 0.76 SLC40A1 (0.66) SLC40A1MEN1KMT2ANFKBIARELA
SCHEMBL13633852 0.76 SLC40A1 (0.67) SLC40A1MEN1KMT2ANFKBIARELA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8470821-B2 PDE4B inhibitors and uses therefor PLEXXIKON INC. (US) 2013-06-25 US disclosed
US-8470821-B2 PDE4B inhibitors and uses therefor PLEXXIKON INC. (US) 2013-06-25 US disclosed
US-20090286793-A1 PDE4B INHIBITORS AND USES THEREFOR PLEXXIKON, INC. 2009-11-19 US disclosed
US-20090286793-A1 PDE4B INHIBITORS AND USES THEREFOR PLEXXIKON, INC. 2009-11-19 US disclosed
US-7585859-B2 PDE4B inhibitors and uses therefor PLEXXIKON, INC. (US) 2009-09-08 US disclosed
US-7585859-B2 PDE4B inhibitors and uses therefor PLEXXIKON, INC. (US) 2009-09-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090286793-A1 PDE4B INHIBITORS AND USES THEREFOR PDE4B, PDE7B, PDE4A SLC40A1 4638/4885MEN1 2737/4885KMT2A 2234/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.