SCHEMBL13635355

SCHEMBL13635355

CCCCNC(=O)c1ccc2[nH]nc(-c3ccc4ccccc4c3)c2c1OC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
LMNA P02545 2/20 0.42
HDAC3 O15379 2/20 0.42
HDAC1 Q13547 2/20 0.42
HDAC2 Q92769 2/20 0.42
HDAC4 P56524 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
HDAC9 Q9UKV0 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42
DRD2 P14416 2/20 0.41
DRD3 P35462 2/20 0.41
KDR P35968 2/20 0.41
CDK4 P11802 1/20 0.41
CCNA2 P20248 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13198250 0.92 HDAC6 (0.50) LMNAHDAC3HDAC1HDAC2HDAC4
SCHEMBL4331810 0.89 KDR (0.42) KDM4EALDH1A1LMNAHDAC3HDAC1
SCHEMBL4348178 0.88 LMNA (0.45) MAPTLMNAHDAC3HDAC1HDAC2
SCHEMBL2864362 0.84 GSK3B (0.44) DRD2KDRCDK4CCNA2CCND1
SCHEMBL4335936 0.84 BRD4 (0.47) ALDH1A1MAPTKDRCDK4CCNA2
SCHEMBL4335955 0.84 RCE1 (0.54) KDM4EALDH1A1LMNATSHRNPC1
SCHEMBL2864594 0.83 KDR (0.47) KDRCDK4CCNA2CCND1CDK2
SCHEMBL4334496 0.83 MEN1 (0.41) DRD2DRD3KDRCDK4CCNA2
SCHEMBL4341067 0.83 RAB9A (0.46) KDM4EALDH1A1MAPTLMNATSHR
SCHEMBL2856935 0.83 SMN1; SMN2 (0.54) KDM4EALDH1A1MAPTHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1380576-B1 1H-INDAZOLE COMPOUNDS INHIBITING JNK EISAI R&D MAN CO LTD (JP) 2009-11-25 EP disclosed