SCHEMBL13635754

SCHEMBL13635754

O=C(NCC1C=COC1)c1cc(F)c2[nH]nc(-c3cccc(F)c3)c2c1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 1/20 0.37
GSK3B P49841 7/20 0.36
CYP1A2 P05177 1/20 0.36
GAA P10253 1/20 0.36
CYP2C9 P11712 1/20 0.36
HPGD P15428 1/20 0.36
CYP2C19 P33261 1/20 0.36
MAP2K4 P45985 2/20 0.35
DYRK1A Q13627 1/20 0.35
KLKB1 P03952 2/20 0.34
GSK3A P49840 1/20 0.34
PTAFR P25105 1/20 0.34
KCNH2 Q12809 5/20 0.33
OPRM1 P35372 1/20 0.33
CCNA2 P20248 1/20 0.33
CDK2 P24941 1/20 0.33
CCNA1 P78396 1/20 0.33
MAP2K7 O14733 1/20 0.33
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13635757 0.88 ITK (0.34) GSK3BKCNH2
SCHEMBL2866665 0.84 GABRA5 (0.48) GABRA5GSK3BCYP1A2GAACYP2C9
SCHEMBL4331604 0.80 HPGD (0.61) GSK3BCYP1A2GAACYP2C9HPGD
SCHEMBL4332657 0.80 HPGD (0.61) GSK3BCYP1A2GAACYP2C9HPGD
SCHEMBL2865663 0.77 DYRK1A (0.48) GABRA5GSK3BMAP2K4DYRK1AGSK3A
SCHEMBL4345594 0.76 HPGD (0.42) GABRA5HPGDTP53
SCHEMBL4327002 0.76 HPGD (0.58) GAAHPGD
SCHEMBL4334573 0.76 TTK (0.55) GAAHPGD
SCHEMBL4334999 0.76 TP53 (0.41) CYP1A2HPGDMAP2K4PTAFRTP53
SCHEMBL4334327 0.75 PARP1 (0.43) HPGDKLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1380576-B1 1H-INDAZOLE COMPOUNDS INHIBITING JNK EISAI R&D MAN CO LTD (JP) 2009-11-25 EP disclosed