SCHEMBL13636201

SCHEMBL13636201

O=C(CCc1ccc(O)c(O)c1)N1CCN(C2CCCC2)CC1

nearest known ligand 0.63

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.63
KMT2A Q03164 2/20 0.63
TSHR P16473 1/20 0.63
L3MBTL3 Q96JM7 1/20 0.54
KDM4E B2RXH2 3/20 0.53
HRH3 Q9Y5N1 7/20 0.51
POLB P06746 1/20 0.47
MAPT P10636 1/20 0.47
CCR5 P51681 1/20 0.46
ROCK2 O75116 2/20 0.45
TACR1 P25103 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13090092 0.90 L3MBTL3 (0.64) ALDH1A1KMT2ATSHRL3MBTL3POLB
SCHEMBL9345400 0.83 NPC1 (0.61) ALDH1A1KMT2APOLBMAPT
SCHEMBL9350110 0.82 NPC1 (0.59) ALDH1A1KMT2APOLBMAPT
SCHEMBL4377238 0.81 KMT2A (0.71) ALDH1A1KMT2ATSHRL3MBTL3KDM4E
SCHEMBL4378534 0.81 KMT2A (0.62) ALDH1A1KMT2ATSHRL3MBTL3KDM4E
SCHEMBL4375187 0.80 KMT2A (0.73) ALDH1A1KMT2ATSHRL3MBTL3
SCHEMBL4379319 0.80 KMT2A (0.64) ALDH1A1KMT2ATSHRL3MBTL3KDM4E
SCHEMBL9346536 0.80 IAPP (0.53) KMT2ATSHRMAPTROCK2
SCHEMBL13636198 0.79 ALDH1A1 (0.56) ALDH1A1KMT2ATSHRL3MBTL3KDM4E
SCHEMBL4383272 0.79 ALDH1A1 (0.98) ALDH1A1KMT2ATSHRL3MBTL3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1421071-B1 SUBSTITUTED PIPERAZINE AND DIAZEPANE DERIVAIVES AS HISTAMINE H3 RECEPTOR MODULATORS HIGH POINT PHARMACEUTICALS LLC (US) 2009-11-18 EP disclosed