SCHEMBL13638251

SCHEMBL13638251

COc1ccc2cccc(CC[C@H]3CC[C@H](NCc4cnc5c(c4)NC(=O)CS5)CC3)c2n1

nearest known ligand 0.43

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 7/20 0.43
MTNR1B P49286 7/20 0.43
KCNH2 Q12809 4/20 0.39
SIRT2 Q8IXJ6 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13633343 0.88 KCNH2 (0.46) MTNR1AMTNR1BKCNH2SIRT2
SCHEMBL3572910 0.88 KCNH2 (0.46) MTNR1AMTNR1BKCNH2SIRT2
SCHEMBL3572912 0.81 MTNR1A (0.38) MTNR1AMTNR1BKCNH2
SCHEMBL20679509 0.79 MTNR1A (0.43) MTNR1AMTNR1BKCNH2
SCHEMBL6668585 0.74 KCNH2 (0.58) KCNH2
Hydrochloric Acid SCHEMBL5745883 0.73 KCNH2 (0.61) KCNH2
SCHEMBL5263873 0.72 KCNH2 (0.52) KCNH2
SCHEMBL5253266 0.72 KCNH2 (0.59) KCNH2
SCHEMBL5253262 0.72 KCNH2 (0.59) KCNH2
SCHEMBL5253263 0.72 KCNH2 (0.59) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7622481-B2 Antibacterial compounds GLAXO GROUP LIMITED (GB) 2009-11-24 US disclosed