SCHEMBL13633343

SCHEMBL13633343

COc1ccc2cccc(CC[C@]3(O)CC[C@@H](NCc4cnc5c(c4)NC(=O)CS5)CC3)c2n1

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.46
MTNR1A P48039 8/20 0.41
MTNR1B P49286 8/20 0.41
SIRT2 Q8IXJ6 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3572910 1.00 KCNH2 (0.46) KCNH2MTNR1AMTNR1BSIRT2
SCHEMBL13638251 0.88 MTNR1A (0.43) KCNH2MTNR1AMTNR1BSIRT2
SCHEMBL3572912 0.87 MTNR1A (0.38) KCNH2MTNR1AMTNR1B
SCHEMBL13407409 0.80 KCNH2 (0.44) KCNH2MTNR1AMTNR1B
SCHEMBL3574972 0.80 KCNH2 (0.44) KCNH2MTNR1AMTNR1B
SCHEMBL6102949 0.78 KCNH2 (0.39) KCNH2MTNR1AMTNR1BSIRT2
SCHEMBL14341402 0.76 KCNH2 (0.68) KCNH2
SCHEMBL20679509 0.76 MTNR1A (0.43) KCNH2MTNR1AMTNR1B
SCHEMBL6195137 0.74 KCNH2 (0.46) KCNH2MTNR1AMTNR1B
SCHEMBL3582737 0.73 KCNH2 (0.54) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7622481-B2 Antibacterial compounds GLAXO GROUP LIMITED (GB) 2009-11-24 US disclosed
EP-1537123-B1 AMINO-SUBSTITUTED CYCLOHEXANE DERIVATIVES FOR THE TREATMENT OF BACTERIAL INFECTIONS GLAXO GROUP LTD (GB) 2009-04-29 EP disclosed