SCHEMBL13638313

SCHEMBL13638313

C=C1CC(Nc2nccc(-c3ccc(CCCCN)cc3)n2)CC(C)(C)N1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 14/20 0.39
CHUK O15111 2/20 0.37
MAPK8 P45983 3/20 0.36
AKT2 P31751 1/20 0.34
AURKA O14965 1/20 0.34
TTK P33981 1/20 0.34
AURKB Q96GD4 1/20 0.34
INCENP Q9NQS7 1/20 0.34
ROCK2 O75116 3/20 0.34
MAPK9 P45984 2/20 0.34
MAPK10 P53779 2/20 0.34
MAPK11 Q15759 1/20 0.34
MAPK14 Q16539 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13638312 0.97 IKBKB (0.39) IKBKBCHUKMAPK8AKT2AURKA
SCHEMBL13638679 0.94 IKBKB (0.41) IKBKBCHUKMAPK8AURKATTK
SCHEMBL13638438 0.90 IKBKB (0.39) IKBKBCHUKMAPK8ROCK2MAPK9
SCHEMBL13638538 0.88 IKBKB (0.38) IKBKBCHUKMAPK8MAPK11MAPK14
SCHEMBL4492944 0.87 IKBKB (0.42) IKBKBCHUKMAPK8AURKATTK
SCHEMBL13638591 0.87 IKBKB (0.37) IKBKBCHUKMAPK8AURKATTK
SCHEMBL13638532 0.87 IKBKB (0.39) IKBKBCHUKMAPK8AURKATTK
SCHEMBL13638590 0.86 ROCK2 (0.38) IKBKBCHUKMAPK8AURKATTK
SCHEMBL13638437 0.85 IKBKB (0.39) IKBKBCHUKMAPK8MAPK9MAPK10
SCHEMBL13638531 0.85 SYK (0.43) IKBKBCHUKMAPK8ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7615562-B2 Such as 2-methyl-4-{5-[2-(2,2,6,6-tetramethyl-piperidin-4-ylamino)-pyrimidin-4-yl]-thiophen-2-yl}-butan-2-ol; tumor necrosis factor inhibitors; immunosuppressants; antiinflammatory agents NOVARTIS AG (CH) 2009-11-10 US disclosed