SCHEMBL13638531

SCHEMBL13638531

C=C1CC(Nc2nccc(-c3ccc(CCC(=O)O)cc3)n2)CC(C)(C)N1

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SYK P43405 5/20 0.43
IKBKB O14920 9/20 0.37
HDAC8 Q9BY41 5/20 0.37
MAPK8 P45983 1/20 0.36
HDAC6 Q9UBN7 2/20 0.36
CHUK O15111 1/20 0.36
ROCK2 O75116 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13638482 0.93 IKBKB (0.37) SYKIKBKBHDAC8MAPK8HDAC6
SCHEMBL13638590 0.92 ROCK2 (0.38) SYKIKBKBHDAC8MAPK8HDAC6
SCHEMBL13638534 0.91 JAK2 (0.39) SYKIKBKBHDAC8MAPK8HDAC6
SCHEMBL13638438 0.88 IKBKB (0.39) IKBKBHDAC8MAPK8HDAC6CHUK
SCHEMBL13638540 0.87 IKBKB (0.39) IKBKBHDAC8MAPK8HDAC6ROCK2
SCHEMBL13638679 0.87 IKBKB (0.41) IKBKBMAPK8CHUK
SCHEMBL4482129 0.87 SYK (0.46) SYKIKBKBHDAC8MAPK8ROCK2
SCHEMBL13638312 0.86 IKBKB (0.39) IKBKBMAPK8CHUKROCK2
SCHEMBL13638437 0.85 IKBKB (0.39) IKBKBHDAC8MAPK8CHUK
SCHEMBL13638536 0.85 IKBKB (0.37) IKBKBHDAC8MAPK8CHUK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7615562-B2 Such as 2-methyl-4-{5-[2-(2,2,6,6-tetramethyl-piperidin-4-ylamino)-pyrimidin-4-yl]-thiophen-2-yl}-butan-2-ol; tumor necrosis factor inhibitors; immunosuppressants; antiinflammatory agents NOVARTIS AG (CH) 2009-11-10 US disclosed