SCHEMBL13638407

SCHEMBL13638407

C#CC(C)(C)OC(=O)CC(NC(=O)C(CC)n1ccc2ccc(Cl)cc2c1=O)C(=O)COc1c(F)c(F)cc(F)c1F

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 18/20 0.38
CASP6 P55212 8/20 0.38
CASP8 Q14790 8/20 0.38
CASP1 P29466 2/20 0.37
CASP7 P55210 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3582995 1.00 CASP3 (0.38) CASP3CASP6CASP8CASP1CASP7
SCHEMBL8320800 0.92 CASP1 (0.39) CASP3CASP6CASP8CASP1CASP7
SCHEMBL12046989 0.92 CASP1 (0.39) CASP3CASP6CASP8CASP1CASP7
SCHEMBL12046795 0.91 CASP1 (0.39) CASP3CASP6CASP8CASP1CASP7
SCHEMBL12046805 0.90 CASP1 (0.38) CASP3CASP6CASP8CASP1CASP7
SCHEMBL3582997 0.90 CASP3 (0.37) CASP3CASP6CASP8CASP1CASP7
SCHEMBL3587580 0.89 CASP1 (0.41) CASP3CASP6CASP8CASP1CASP7
SCHEMBL3587583 0.89 CASP1 (0.41) CASP3CASP6CASP8CASP1CASP7
SCHEMBL8315069 0.89 CASP1 (0.41) CASP3CASP6CASP8CASP1CASP7
SCHEMBL3587578 0.89 CASP1 (0.41) CASP3CASP6CASP8CASP1CASP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612091-B2 Caspase inhibitors and uses thereof VERTEX PHARMACEUTICALS INCORPORATED (US) 2009-11-03 US disclosed