SCHEMBL13638526

SCHEMBL13638526

C=C1CC(Nc2ncc(C)c(-c3cc4ccc(OC)cc4s3)n2)CC(C)(C)N1

nearest known ligand 0.32

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EIF2AK2 P19525 1/20 0.32
KCNH2 Q12809 1/20 0.32
FGFR1 P11362 1/20 0.32
FGFR4 P22455 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.31
CHRNA7 P36544 3/20 0.31
KDR P35968 1/20 0.31
PLK1 P53350 1/20 0.31
AXL P30530 1/20 0.31
MERTK Q12866 1/20 0.31
HPGDS O60760 1/20 0.30
SNCA P37840 1/20 0.30
IGF1R P08069 1/20 0.30
MAPK6 Q16659 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3476836 0.88 KCNH2 (0.42) EIF2AK2KCNH2FGFR1FGFR4CHRNA7
SCHEMBL13638316 0.87 KCNH2 (0.44) KCNH2MERTK
SCHEMBL13638581 0.86 EIF2AK2 (0.40) EIF2AK2KCNH2FGFR1FGFR4
SCHEMBL13638475 0.84 ADRB2 (0.35)
SCHEMBL13638524 0.76 KCNH2 (0.33) EIF2AK2KCNH2
SCHEMBL14612852 0.76 KCNH2 (0.39) KCNH2MERTK
SCHEMBL13638308 0.76 KCNH2 (0.34) EIF2AK2KCNH2SMN1; SMN2
SCHEMBL3476962 0.74 KCNH2 (0.58) KCNH2MERTK
SCHEMBL13638505 0.74 JUN (0.31)
SCHEMBL13638661 0.73 RPS6KB2 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7615562-B2 Such as 2-methyl-4-{5-[2-(2,2,6,6-tetramethyl-piperidin-4-ylamino)-pyrimidin-4-yl]-thiophen-2-yl}-butan-2-ol; tumor necrosis factor inhibitors; immunosuppressants; antiinflammatory agents NOVARTIS AG (CH) 2009-11-10 US disclosed