SCHEMBL13638540

SCHEMBL13638540

C=C1CC(Nc2nccc(-c3ccc(CC(C)=O)cc3)n2)CC(C)(C)N1

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 10/20 0.39
HDAC8 Q9BY41 5/20 0.38
MAPK8 P45983 2/20 0.38
WNT3A P56704 1/20 0.37
HDAC6 Q9UBN7 1/20 0.36
ROCK2 O75116 3/20 0.36
MAPK9 P45984 1/20 0.35
MAPK10 P53779 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13638482 0.91 IKBKB (0.37) IKBKBHDAC8MAPK8HDAC6ROCK2
SCHEMBL13638531 0.87 SYK (0.43) IKBKBHDAC8MAPK8HDAC6ROCK2
SCHEMBL13638592 0.87 IKBKB (0.41) IKBKBHDAC8MAPK8ROCK2MAPK9
SCHEMBL13638590 0.86 ROCK2 (0.38) IKBKBHDAC8MAPK8HDAC6ROCK2
SCHEMBL4484136 0.86 IKBKB (0.42) IKBKBHDAC8MAPK8WNT3AROCK2
SCHEMBL13638438 0.86 IKBKB (0.39) IKBKBHDAC8MAPK8HDAC6ROCK2
SCHEMBL13638534 0.85 JAK2 (0.39) IKBKBHDAC8MAPK8HDAC6ROCK2
SCHEMBL13638536 0.85 IKBKB (0.37) IKBKBHDAC8MAPK8MAPK9MAPK10
SCHEMBL13638440 0.85 IKBKB (0.43) IKBKBHDAC8MAPK8MAPK9MAPK10
SCHEMBL13638679 0.85 IKBKB (0.41) IKBKBMAPK8MAPK9MAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7615562-B2 Such as 2-methyl-4-{5-[2-(2,2,6,6-tetramethyl-piperidin-4-ylamino)-pyrimidin-4-yl]-thiophen-2-yl}-butan-2-ol; tumor necrosis factor inhibitors; immunosuppressants; antiinflammatory agents NOVARTIS AG (CH) 2009-11-10 US disclosed