SCHEMBL13638589

SCHEMBL13638589

C=C1CC(Nc2nccc(-n3cc(C(C)=O)c4ccccc43)n2)CC(C)(C)N1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 12/20 0.42
MAPK9 P45984 6/20 0.41
MAPK10 P53779 5/20 0.41
CDK2 P24941 2/20 0.40
JUN P05412 1/20 0.40
MKNK1 Q9BUB5 8/20 0.40
MKNK2 Q9HBH9 7/20 0.40
CYP2C9 P11712 1/20 0.39
CCNE1 P24864 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13638311 0.92 MAPK8 (0.47) MAPK8MAPK9MAPK10CDK2JUN
SCHEMBL4478671 0.88 MAPK8 (0.44) MAPK8MAPK9MAPK10CDK2JUN
SCHEMBL13638681 0.83 MAPK8 (0.48) MAPK8MAPK9MAPK10
SCHEMBL13638441 0.80 MAPK8 (0.58) MAPK8MAPK9MAPK10CDK2JUN
SCHEMBL4488358 0.80 MAPK8 (0.49) MAPK8MAPK9MAPK10CDK2JUN
SCHEMBL13638543 0.77 MAPK8 (0.47) MAPK8MAPK9MAPK10MKNK1
SCHEMBL13638545 0.74 CCNB2 (0.48) CDK2MKNK1MKNK2
SCHEMBL14193741 0.71 MAPK8 (0.55) MAPK8MAPK9MAPK10CDK2JUN
SCHEMBL13638593 0.71 ROCK1 (0.49) MAPK8MAPK9MAPK10CDK2JUN
SCHEMBL5090355 0.71 MAPK8 (0.62) MAPK8MAPK9MAPK10CDK2MKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7615562-B2 Such as 2-methyl-4-{5-[2-(2,2,6,6-tetramethyl-piperidin-4-ylamino)-pyrimidin-4-yl]-thiophen-2-yl}-butan-2-ol; tumor necrosis factor inhibitors; immunosuppressants; antiinflammatory agents NOVARTIS AG (CH) 2009-11-10 US disclosed