SCHEMBL13638760

SCHEMBL13638760

COc1cc(N)cc(Oc2c(Cl)ccc(CNC(=O)c3[nH]c(N)nc3Cl)c2F)c1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGES O14684 10/20 0.37
CHRM4 P08173 2/20 0.35
RORC P51449 1/20 0.35
WDR5 P61964 2/20 0.34
ROCK2 O75116 1/20 0.34
ROCK1 Q13464 1/20 0.34
BCHE P06276 1/20 0.34
ACHE P22303 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
KMT2A Q03164 1/20 0.34
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
MEP1B Q16820 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13982372 0.92 PTGES (0.37) PTGESCHRM4RORCWDR5ROCK2
SCHEMBL3029925 0.92 CYP3A4 (0.43) PTGESCHRM4RORCWDR5ROCK2
SCHEMBL13982340 0.91 PTGES (0.35) PTGESCYP3A4
SCHEMBL13982447 0.88 PTGES (0.39) PTGESRORC
Trifluoroacetic Acid SCHEMBL13560564 0.87 CYP3A4 (0.40) PTGESRORCWDR5KDM4EMEN1
SCHEMBL13982463 0.87 PTGES (0.38) PTGESRORCROCK2ROCK1CYP3A4
SCHEMBL13982440 0.86 PTGES (0.36) PTGES
SCHEMBL13982369 0.86 RORC (0.35) PTGESCHRM4RORCWDR5ROCK2
SCHEMBL13982357 0.86 EPHX2 (0.32) PTGESRORCROCK2ROCK1CYP3A4
SCHEMBL13982434 0.84 PTGES (0.35) PTGESALDH1A1KMT2ACYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8304419-B2 Chemical compounds GLAXOSMITHKLINE LLC (US) 2012-11-06 US disclosed
WO-2008154271-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-18 WO disclosed