SCHEMBL13639808

SCHEMBL13639808

Cc1cc(-c2cn[nH]c(=O)c2)cc(C)c1OCCCN1CCCC1

nearest known ligand 0.67

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 6/20 0.67
ALDH1A1 P00352 1/20 0.50
HRH3 Q9Y5N1 6/20 0.49
KCNH2 Q12809 1/20 0.49
BRD4 O60885 1/20 0.43
IL17A Q16552 1/20 0.43
HTR1A P08908 1/20 0.41
HTR2A P28223 1/20 0.41
HTR7 P34969 1/20 0.41
KDM4E B2RXH2 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14319716 0.83 HTR3A (0.76) HTR3AHRH3KCNH2
SCHEMBL1375386 0.82 HTR3A (0.78) HTR3AHRH3KCNH2
SCHEMBL14308933 0.81 HTR3A (0.98) HTR3AHRH3KCNH2
SCHEMBL10197092 0.80 HTR3A (1.00) HTR3AHRH3KCNH2
SCHEMBL1373384 0.71 HRH3 (0.72) HTR3AHRH3KCNH2
SCHEMBL1373387 0.71 HRH3 (0.72) HTR3AHRH3KCNH2
SCHEMBL10260801 0.69 HTR3A (0.71) HTR3AHRH3
SCHEMBL12017517 0.69 HRH3 (0.67) HTR3AHRH3KCNH2
SCHEMBL24163014 0.69 L3MBTL1 (0.71) ALDH1A1HRH3HTR1AHTR2AHTR7
SCHEMBL1373734 0.68 HRH3 (0.82) HTR3AHRH3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2069312-B1 PYRIDIZINONE DERIVATIVES CEPHALON INC (US) 2012-11-07 EP disclosed