SCHEMBL13639810

SCHEMBL13639810

C[C@H](COc1ccc(-c2cn[nH]c(=O)c2)cc1)CN1CCCC1

nearest known ligand 0.98

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 9/20 0.98
HTR3A P46098 6/20 0.65
KCNH2 Q12809 3/20 0.53
ADORA2A P29274 1/20 0.42
ATM Q13315 1/20 0.41
KMT2A Q03164 1/20 0.41
SIGMAR1 Q99720 2/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1376239 0.99 HRH3 (1.00) HRH3HTR3AKCNH2ADORA2AATM
SCHEMBL1375082 0.99 HRH3 (1.00) HRH3HTR3AKCNH2ADORA2AATM
SCHEMBL1375085 0.99 HRH3 (1.00) HRH3HTR3AKCNH2ADORA2AATM
SCHEMBL1376743 0.84 HRH3 (1.00) HRH3HTR3AKCNH2
SCHEMBL1372936 0.84 HRH3 (1.00) HRH3HTR3AKCNH2
SCHEMBL1372932 0.84 HRH3 (1.00) HRH3HTR3AKCNH2
SCHEMBL14308933 0.80 HTR3A (0.98) HRH3HTR3AKCNH2
SCHEMBL10197092 0.79 HTR3A (1.00) HRH3HTR3AKCNH2
SCHEMBL10267647 0.78 HRH3 (0.66) HRH3HTR3AKCNH2KMT2A
SCHEMBL13639811 0.76 HRH3 (0.60) HRH3HTR3AKCNH2CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2069312-B1 PYRIDIZINONE DERIVATIVES CEPHALON INC (US) 2012-11-07 EP disclosed