SCHEMBL13650897

SCHEMBL13650897

N=c1sc2c(n1CC(=O)c1cccc(F)c1)CCCC2

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.64
SMN1; SMN2 Q16637 4/20 0.64
KMT2A Q03164 3/20 0.64
CYP1A1 P04798 2/20 0.64
CYP1B1 Q16678 2/20 0.64
ALDH1A1 P00352 2/20 0.64
MEN1 O00255 2/20 0.64
TSHR P16473 2/20 0.64
TP53 P04637 1/20 0.64
CYP3A4 P08684 1/20 0.64
ALOX15 P16050 1/20 0.64
MAPK1 P28482 1/20 0.64
HSD17B10 Q99714 1/20 0.64
HDAC6 Q9UBN7 1/20 0.64
RXFP1 Q9HBX9 1/20 0.41
GRIN2B Q13224 1/20 0.39
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37
CTNNB1 P35222 2/20 0.37
WNT3A P56704 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL29440222 0.99 CYP1A1 (0.65) MAPTSMN1; SMN2KMT2ACYP1A1CYP1B1
Bromide SCHEMBL22749637 0.99 CYP1A1 (0.65) MAPTSMN1; SMN2KMT2ACYP1A1CYP1B1
Bromide SCHEMBL22749635 0.98 MAPT (0.61) MAPTSMN1; SMN2KMT2ACYP1A1CYP1B1
SCHEMBL22761718 0.86 ALDH1A1 (0.64) MAPTSMN1; SMN2KMT2ACYP1A1CYP1B1
SCHEMBL22761628 0.86 MEN1 (0.64) MAPTSMN1; SMN2KMT2ACYP1A1CYP1B1
SCHEMBL4942836 0.85 ALDH1A1 (0.77) MAPTSMN1; SMN2KMT2ACYP1A1CYP1B1
SCHEMBL4941971 0.85 ALDH1A1 (0.77) MAPTSMN1; SMN2KMT2ACYP1A1CYP1B1
Bromide SCHEMBL4796807 0.85 CYP1A1 (0.75) MAPTSMN1; SMN2KMT2ACYP1A1CYP1B1
Bromide SCHEMBL22749445 0.85 CYP1A1 (0.65) MAPTSMN1; SMN2KMT2ACYP1A1CYP1B1
Bromide SCHEMBL22749448 0.85 CYP1A1 (0.65) MAPTSMN1; SMN2KMT2ACYP1A1CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020247336-A1 PIFITHRIN ANALOGUES AND METHODS OF TREATING RETT SYNDROME THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2020-12-10 WO disclosed
US-7601846-B2 Compounds having activity as inhibitors of apoptosis THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2009-10-13 US disclosed