SCHEMBL13655518

SCHEMBL13655518

Cc1ccc2cc(I)[nH]c2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 1/20 0.52
DDO Q99489 1/20 0.52
MAPT P10636 1/20 0.49
RXFP1 Q9HBX9 1/20 0.49
CA12 O43570 1/20 0.47
CA9 Q16790 1/20 0.47
ALDH1A1 P00352 4/20 0.45
ITK Q08881 3/20 0.45
KDM4E B2RXH2 3/20 0.45
HSD17B10 Q99714 2/20 0.45
CYP1A2 P05177 3/20 0.44
CYP2A6 P11509 2/20 0.44
FLT3 P36888 2/20 0.42
HIF1A Q16665 2/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
GRIN2D O15399 1/20 0.41
GRIN3B O60391 1/20 0.41
GRIN1 Q05586 1/20 0.41
GRIN2A Q12879 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20280559 0.83 LOXL2 (0.53) DAOMAPTCA12CA9ALDH1A1
SCHEMBL890079 0.77 DAO (0.55) DAODDOMAPTRXFP1CA12
SCHEMBL30807019 0.77 DAO (0.55) DAODDOMAPTRXFP1CA12
SCHEMBL27957027 0.74 DAO (0.52) DAODDOMAPTRXFP1CA12
SCHEMBL8959176 0.74 AOC3 (0.54) DAODDOMAPTRXFP1CA12
SCHEMBL8288035 0.74 DAO (0.52) DAODDOMAPTRXFP1CA12
SCHEMBL12777915 0.74
SCHEMBL28798245 0.74 DAO (0.52) DAOALDH1A1HSD17B10GRIN2DGRIN3B
SCHEMBL12778114 0.74 CA2 (0.54) MAPTRXFP1ALDH1A1ITKKDM4E
SCHEMBL28024614 0.71 MAPT (0.51) DAODDOMAPTRXFP1CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1381366-B9 INDOLE, AZAINDOLE AND RELATED HETEROCYCLIC AMIDOPIPERAZINE DERIVATIVES BRISTOL MYERS SQUIBB CO (US) 2009-10-21 EP disclosed
EP-1381366-B1 INDOLE, AZAINDOLE AND RELATED HETEROCYCLIC AMIDOPIPERAZINE DERIVATIVES BRISTOL MYERS SQUIBB CO (US) 2009-04-22 EP disclosed