Prulifloxacin

Prulifloxacin

SCHEMBL136641

Cc1oc(=O)oc1CN1CCN(c2cc3c(cc2F)c(=O)c(C(=O)O)c2n3[C@@H](C)S2)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

gyrAgyrBparCparE

The experimentally established mechanism targets of Prulifloxacin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 1.00
PRKD3 O94806 1/20 0.46
PIM1 P11309 1/20 0.46
GSK3A P49840 1/20 0.46
GSK3B P49841 1/20 0.46
IRAK1 P51617 1/20 0.46
RPS6KA3 P51812 1/20 0.46
DYRK1A Q13627 1/20 0.46
PIM3 Q86V86 1/20 0.46
CSNK1G3 Q9Y6M4 1/20 0.46
ALDH1A1 P00352 7/20 0.41
KDM4E B2RXH2 6/20 0.41
HSD17B10 Q99714 5/20 0.41
HPGD P15428 5/20 0.41
MAPT P10636 1/20 0.41
DRD3 P35462 1/20 0.38
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
BRD4 O60885 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Prulifloxacin SCHEMBL13896543 1.00 LMNA (1.00) LMNAPRKD3PIM1GSK3AGSK3B
Prulifloxacin SCHEMBL1650794 1.00 LMNA (1.00) LMNAPRKD3PIM1GSK3AGSK3B
Prulifloxacin SCHEMBL1699755 1.00 LMNA (1.00) LMNAPRKD3PIM1GSK3AGSK3B
Prulifloxacin SCHEMBL29540773 1.00 LMNA (1.00) LMNAPRKD3PIM1GSK3AGSK3B
Prulifloxacin SCHEMBL7060281 1.00 LMNA (1.00) LMNAPRKD3PIM1GSK3AGSK3B
Prulifloxacin SCHEMBL13822719 0.99 LMNA (0.98) LMNAPRKD3PIM1GSK3AGSK3B
Prulifloxacin SCHEMBL28660626 0.99 LMNA (0.98) LMNAPRKD3PIM1GSK3AGSK3B
Prulifloxacin SCHEMBL9673724 0.99 LMNA (0.98) LMNAPRKD3PIM1GSK3AGSK3B
Prulifloxacin SCHEMBL1231520 0.99 LMNA (0.98) LMNAPRKD3PIM1GSK3AGSK3B
Prulifloxacin SCHEMBL9674383 0.96 LMNA (0.92) LMNAPRKD3PIM1GSK3AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3822 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12624057-B2 Bisphosphonate quinolone conjugates and uses thereof BIOVINC, LLC (US) 2026-05-12 US claimed
EP-4658376-A1 SKIN CARE COMPOSITIONS Colgate-Palmolive Company (US) 2025-12-10 EP claimed
US-20250346910-A1 METHODS AND COMPOSITIONS TO PREVENT MICROBIAL INFECTION COMMENSE BIO INC (US) 2025-11-13 US claimed
US-20250262167-A1 COMPOUNDS, TARGETS AND PATHWAYS FOR MACROPHAGE MODULATION MASSACHUSETTS INSTITUTE OF TECHNOLOGY 2025-08-21 US claimed
CN-120131953-A Targeted nano-drug with sonodynamic activity, and preparation method and application thereof 中山大学·深圳 2025-06-13 CN claimed
EP-4554627-A1 INHALABLE FORMULATION FOR USE IN THE TREATMENT OF BACTERIAL LUNG INFECTIONS Solmic Biotech GmbH (DE) 2025-05-21 EP claimed
EP-4554939-A1 PCSK9 INHIBITORS AND METHODS OF USE THEREOF Astrazeneca AB (SE) 2025-05-21 EP claimed
US-20250144088-A1 INHALABLE FORMULATION FOR USE IN THE TREATMENT OF BACTERIAL LUNG INFECTIONS Solmic Biotech GmbH (DE) 2025-05-08 US claimed
CN-119875972-A Methods and compositions for preventing microbial infection 比奥普来克斯有限公司 2025-04-25 CN claimed
WO-2025080590-A1 CO-CRYSTALLIZATION OF ACTIVES WITH SACCHARIDE-BASED MOLECULAR FRAMEWORKS SCIENTIFIC HORIZONS CONSULTING LLC (US) 2025-04-17 WO claimed
US-20060018933-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 US claimed
US-20060018934-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 US claimed
CN-1704419-A Process for synthesis of prulifloxacin and its pharmaceutical composition HARBIN JIANDI MEDICINE TECHNOL (CN) 2005-12-07 CN claimed
CN-1668598-A Use of chemotherapeutic agents SCHULZ & SCHLIMBACH GBR (DE) 2005-09-14 CN claimed
CN-1557314-A Prulifloxacin water-soluble salt and its injection formulation 魏雪纹 2004-12-29 CN claimed
EP-1408034-A1 Use of Quinoline derivatives as antibacterial agents Schulz & Schlimbach GbR (DE) 2004-04-14 EP claimed
CN-1478781-A Preparation method of prolisaxin 高 杨 2004-03-03 CN claimed
EP-1244434-A2 USE OF CHEMOTHERAPEUTIC AGENTS Schulz, Hans-Herrmann (DE) 2002-10-02 EP claimed
WO-2001045679-A2 USE OF CHEMOTHERAPEUTIC AGENTS FOR TOPICAL TREATMENT SCHULZ HANS HERRMANN (DE) 2001-06-28 WO claimed
WO-2000001365-A1 PROLONGED RELEASE OPHTHALMIC COMPOSITIONS CONTAINING A FLUOROQUINOLONE Leo Pharmaceutical Products Ltd. A/S (Løvens Kemiske Fabrik Produktionsaktieselskab) (DK) 2000-01-13 WO claimed