Prulifloxacin

Prulifloxacin

SCHEMBL1650794

Cc1oc(=O)oc1CN1CCN(c2cc3c(cc2F)c(=O)c(C(=O)O)c2n3C(C)S2)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

gyrAgyrBparCparE

The experimentally established mechanism targets of Prulifloxacin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 1.00
PRKD3 O94806 1/20 0.46
PIM1 P11309 1/20 0.46
GSK3A P49840 1/20 0.46
GSK3B P49841 1/20 0.46
IRAK1 P51617 1/20 0.46
RPS6KA3 P51812 1/20 0.46
DYRK1A Q13627 1/20 0.46
PIM3 Q86V86 1/20 0.46
CSNK1G3 Q9Y6M4 1/20 0.46
ALDH1A1 P00352 7/20 0.41
KDM4E B2RXH2 6/20 0.41
HSD17B10 Q99714 5/20 0.41
HPGD P15428 5/20 0.41
MAPT P10636 1/20 0.41
DRD3 P35462 1/20 0.38
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
BRD4 O60885 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Prulifloxacin SCHEMBL13896543 1.00 LMNA (1.00) LMNAPRKD3PIM1GSK3AGSK3B
Prulifloxacin SCHEMBL1699755 1.00 LMNA (1.00) LMNAPRKD3PIM1GSK3AGSK3B
Prulifloxacin SCHEMBL29540773 1.00 LMNA (1.00) LMNAPRKD3PIM1GSK3AGSK3B
Prulifloxacin SCHEMBL7060281 1.00 LMNA (1.00) LMNAPRKD3PIM1GSK3AGSK3B
Prulifloxacin SCHEMBL136641 1.00 LMNA (1.00) LMNAPRKD3PIM1GSK3AGSK3B
Prulifloxacin SCHEMBL13822719 0.99 LMNA (0.98) LMNAPRKD3PIM1GSK3AGSK3B
Prulifloxacin SCHEMBL28660626 0.99 LMNA (0.98) LMNAPRKD3PIM1GSK3AGSK3B
Prulifloxacin SCHEMBL9673724 0.99 LMNA (0.98) LMNAPRKD3PIM1GSK3AGSK3B
Prulifloxacin SCHEMBL1231520 0.99 LMNA (0.98) LMNAPRKD3PIM1GSK3AGSK3B
Prulifloxacin SCHEMBL9674383 0.96 LMNA (0.92) LMNAPRKD3PIM1GSK3AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 132 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2354144-A1 Crystals of quinolinecarboxylic acid derivative solvate Nippon Shinyaku Co., Ltd. (JP) 2011-08-10 EP claimed
US-7612205-B2 Crystals of quinolinecarboxylic acid derivative solvate NIPPON SHINYAKU CO., LTD. (JP) 2009-11-03 US claimed
EP-1408034-B1 Use of Quinolone and Quinolizinone derivatives as chemotherapeutic agents SCHULZ & SCHLIMBACH GBR (DE) 2007-08-08 EP claimed
US-20070149540-A1 Crystals of quinolinecarboxylic acid derivative solvate NIPPON SHINYAKY CO., LTD. (JP) 2007-06-28 US claimed
EP-1626051-A1 CRYSTALS OF QUINOLINECARBOXYLIC ACID DERIVATIVE SOLVATE Nippon Shinyaku Co., Ltd. (JP) 2006-02-15 EP claimed
EP-0580860-B2 METHOD OF MANUFACTURING SOLID DISPERSION NIPPON SHINYAKU CO LTD (JP) 2004-12-15 EP claimed
EP-1408034-A1 Use of Quinoline derivatives as antibacterial agents Schulz & Schlimbach GbR (DE) 2004-04-14 EP claimed
EP-1244434-A2 USE OF CHEMOTHERAPEUTIC AGENTS Schulz, Hans-Herrmann (DE) 2002-10-02 EP claimed
WO-2001045679-A2 USE OF CHEMOTHERAPEUTIC AGENTS FOR TOPICAL TREATMENT SCHULZ HANS HERRMANN (DE) 2001-06-28 WO claimed
EP-0580860-B1 METHOD OF MANUFACTURING SOLID DISPERSION NIPPON SHINYAKU CO LTD (JP) 1997-10-22 EP claimed
EP-4713056-A1 DEVICE FOR PROVIDING CONTINUED BREATH GUIDANCE, METHOD OF OPERATING AN INHALATION DEVICE, INHALATION DEVICE AND INHALATION DEVICE SYSTEM FOR PROVIDING INHALATION PROCESS/BREATH GUIDING Pari Medical Holding GmbH (DE) 2026-03-25 EP disclosed
EP-4712837-A1 METHOD OF OPERATING AN INHALATION DEVICE, INHALATION DEVICE, INHALATION DEVICE SYSTEM FOR PROVIDING INHALATION PROCESS FEEDBACK AND DEVICE FOR PROVIDING FEEDBACK GUIDANCE Pari Medical Holding GmbH (DE) 2026-03-25 EP disclosed
US-12503718-B2 Biomarker and treatment target for alcoholic hepatitis THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2025-12-23 US disclosed
EP-4659255-A1 MEDICAL EVALUATION METHOD, AEROSOL NEBULIZER AND MEDICAL EVALUATION SYSTEM Pari Medical Holding GmbH (DE) 2025-12-10 EP disclosed
US-12263192-B2 Compositions for management of disorders of the gastrointestinal tract PANTHERYX, INC. (US) 2025-04-01 US disclosed
EP-0665009-A1 CRYSTALLINE CONDITION DISLOCATING METHOD NIPPON SHINYAKU COMPANY, LIMITED (JP) 1995-08-02 EP disclosed
EP-0627218-A1 FAST SOLUBLE TABLET NIPPON SHINYAKU COMPANY, LIMITED (JP) 1994-12-07 EP disclosed
EP-0580861-A1 CAPSULE NIPPON SHINYAKU COMPANY, LIMITED (JP) 1994-02-02 EP disclosed
EP-0580860-A1 METHOD OF MANUFACTURING SOLID DISPERSION NIPPON SHINYAKU COMPANY, LIMITED (JP) 1994-02-02 EP disclosed
EP-0315828-B1 QUINOLINECARBOXYLIC ACID DERIVATIVES NIPPON SHINYAKU COMPANY, LIMITED (JP) 1992-04-08 EP disclosed