SCHEMBL1366633

SCHEMBL1366633

CCOC(=O)c1c[nH]c2ccc(Cl)cc2c1=O

nearest known ligand 0.74

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 4/20 0.74
GABRB2 P47870 4/20 0.74
GABRB1 P18505 3/20 0.73
GABRA3 P34903 3/20 0.73
MEN1 O00255 1/20 0.64
ALDH1A1 P00352 1/20 0.64
TP53 P04637 1/20 0.64
HPGD P15428 1/20 0.64
KMT2A Q03164 1/20 0.64
HSD17B10 Q99714 1/20 0.64
L3MBTL1 Q9Y468 1/20 0.64
NR4A2 P43354 1/20 0.59
CLEC4M Q9H2X3 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30418194 1.00 GABRA1 (0.74) GABRA1GABRB2GABRB1GABRA3MEN1
SCHEMBL5309810 0.91 NR4A2 (0.72) GABRA1GABRB2GABRB1GABRA3MEN1
SCHEMBL27774066 0.90 GABRA1 (0.60) GABRA1GABRB2GABRB1GABRA3MEN1
SCHEMBL30906938 0.90 GABRA1 (0.63) GABRA1GABRB2GABRB1GABRA3MEN1
SCHEMBL30906939 0.90 GABRA1 (0.63) GABRA1GABRB2GABRB1GABRA3MEN1
SCHEMBL7294152 0.90 GABRA1 (0.63) GABRA1GABRB2GABRB1GABRA3MEN1
SCHEMBL28289133 0.88 GABRA1 (0.65) GABRA1GABRB2GABRB1GABRA3MEN1
SCHEMBL30417619 0.86 GABRA1 (0.78) GABRA1GABRB2GABRB1GABRA3MEN1
SCHEMBL7284420 0.86 GABRA1 (0.78) GABRA1GABRB2GABRB1GABRA3MEN1
SCHEMBL7291769 0.85 GABRA1 (1.00) GABRA1GABRB2GABRB1GABRA3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4615523-A1 COMPOUNDS AND THEIR USE KING'S COLLEGE LONDON (GB) 2025-09-17 EP disclosed
WO-2024100095-A1 COMPOUNDS AND THEIR USE KING’S COLLEGE LONDON (GB) 2024-05-16 WO disclosed
WO-2024100095-A1 COMPOUNDS AND THEIR USE KING’S COLLEGE LONDON (GB) 2024-05-16 WO disclosed
CN-109651247-A A kind of green high-efficient synthetic method of carbostyril compound 云南民族大学 2019-04-19 CN disclosed
US-8889706-B2 Soluble mTOR complexes and modulators thereof WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2014-11-18 US disclosed
US-8889706-B2 Soluble mTOR complexes and modulators thereof WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2014-11-18 US disclosed
US-8889706-B2 Soluble mTOR complexes and modulators thereof WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2014-11-18 US disclosed
EP-2350053-B1 Modulators of MTOR Complexes WHITEHEAD BIOMEDICAL INST (US) 2013-12-11 EP disclosed
US-20130072485-A1 SOLUBLE MTOR COMPLEXES AND MODULATORS THEREOF DANA-FARBER CANCER INSTITUTE, INC. (US) 2013-03-21 US disclosed
US-20130072485-A1 SOLUBLE MTOR COMPLEXES AND MODULATORS THEREOF DANA-FARBER CANCER INSTITUTE, INC. (US) 2013-03-21 US disclosed
US-20130072485-A1 SOLUBLE MTOR COMPLEXES AND MODULATORS THEREOF DANA-FARBER CANCER INSTITUTE, INC. (US) 2013-03-21 US disclosed
US-8394818-B2 Soluble mTOR complexes and modulators thereof DANA-FARBER CANCER INSTITUTE, INC. (US) 2013-03-12 US disclosed
US-8394818-B2 Soluble mTOR complexes and modulators thereof DANA-FARBER CANCER INSTITUTE, INC. (US) 2013-03-12 US disclosed
US-8394818-B2 Soluble mTOR complexes and modulators thereof DANA-FARBER CANCER INSTITUTE, INC. (US) 2013-03-12 US disclosed
US-20110288091-A1 SOLUBLE MTOR COMPLEXES AND MODULATORS THEREOF WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2011-11-24 US disclosed
US-20110288091-A1 SOLUBLE MTOR COMPLEXES AND MODULATORS THEREOF WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2011-11-24 US disclosed
US-20110288091-A1 SOLUBLE MTOR COMPLEXES AND MODULATORS THEREOF WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2011-11-24 US disclosed
WO-2010044885-A2 SOLUBLE MTOR COMPLEXES AND MODULATORS THEREOF WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2010-04-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130072485-A1 SOLUBLE MTOR COMPLEXES AND MODULATORS THEREOF MTOR, RICTOR, RPTOR GABRA1 3089/4885GABRB2 2786/4885GABRB1 2799/4885
US-20110288091-A1 SOLUBLE MTOR COMPLEXES AND MODULATORS THEREOF MTOR, RICTOR, RPTOR GABRA1 3089/4885GABRB2 2786/4885GABRB1 2799/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.