SCHEMBL13667451

SCHEMBL13667451

Cc1ncc(C(N)=O)c(-c2ccccc2Cl)n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.53
HSD17B10 Q99714 1/20 0.50
PARP1 P09874 1/20 0.47
ALDH1A1 P00352 2/20 0.46
GRM2 Q14416 1/20 0.42
JAK2 O60674 3/20 0.42
MAP4K4 O95819 1/20 0.42
JAK1 P23458 1/20 0.42
TYK2 P29597 1/20 0.42
GSK3B P49841 1/20 0.42
JAK3 P52333 1/20 0.42
CNR1 P21554 1/20 0.42
IKBKB O14920 2/20 0.42
EPAS1 Q99814 1/20 0.42
KDM4E B2RXH2 1/20 0.42
GAA P10253 1/20 0.42
CYP1A2 P05177 1/20 0.41
MAPT P10636 1/20 0.41
CYP2C9 P11712 1/20 0.41
HPGD P15428 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1016143 0.87 KMT2A (0.58) KMT2AHSD17B10ALDH1A1CNR1CYP1A2
SCHEMBL1013115 0.83 KMT2A (0.51) KMT2AHSD17B10ALDH1A1CNR1EPAS1
SCHEMBL30263390 0.83 SMN1; SMN2 (0.49) KMT2AALDH1A1KDM4ECYP1A2MAPT
SCHEMBL2733287 0.81 ALDH1A1 (0.55) KMT2AALDH1A1KDM4ECYP1A2MAPT
SCHEMBL12575429 0.76 NNMT (0.45) PARP1ALDH1A1JAK2MAP4K4JAK1
SCHEMBL22584044 0.75 NPSR1 (0.46) KMT2APARP1ALDH1A1IKBKBKDM4E
SCHEMBL28062810 0.73 SMN1; SMN2 (0.55) HSD17B10PARP1ALDH1A1JAK2IKBKB
SCHEMBL27480494 0.72 KMT2A (0.43) KMT2AHSD17B10CNR1DPP4
SCHEMBL5189312 0.72 CNR1 (0.48) KMT2AALDH1A1CNR1EPAS1KDM4E
SCHEMBL9589361 0.71 KMT2A (0.53) KMT2AHSD17B10PARP1ALDH1A1GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009130496-A1 SUBSTITUTED PYRIMIDIN-5-CARBOXAMIDES 281 ASTRAZENECA AB (SE) 2009-10-29 WO disclosed