SCHEMBL1366902

SCHEMBL1366902

CC1(O)CCN(Cc2ccc(C(=O)Cn3ncc(OCc4ccccc4)cc3=O)cc2)C1

nearest known ligand 0.82

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 20/20 0.82

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15238893 0.90 MCHR1 (1.00) MCHR1
SCHEMBL4045403 0.88 MCHR1 (0.67) MCHR1
SCHEMBL4050394 0.85 MCHR1 (0.72) MCHR1
SCHEMBL1367999 0.83 MCHR1 (0.66) MCHR1
SCHEMBL1367069 0.82 MCHR1 (0.80) MCHR1
SCHEMBL1368205 0.81 MCHR1 (0.80) MCHR1
SCHEMBL15310571 0.80 MCHR1 (0.77) MCHR1
SCHEMBL1364654 0.80 MCHR1 (0.77) MCHR1
SCHEMBL15310239 0.79 MCHR1 (0.73) MCHR1
SCHEMBL1365170 0.79 MCHR1 (0.76) MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2069327-B1 NEW PYRIDONE DERIVATIVES WITH MCH ANTAGONISTIC ACTIVITY AND MEDICAMENTS COMPRISING THESE COMPOUNDS BOEHRINGER INGELHEIM INT (DE) 2013-10-16 EP claimed
US-8067590-B2 Melanin-concentrating hormone (MCH) receptor antagonists; treating obesity, eating disorders, affective disorders, drug dependency; compounds are amino-functional pyridazin-3-one, 1H-pyridin-2-one or 3H-pyrimidin-4-one BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-11-29 US claimed