SCHEMBL13675242

SCHEMBL13675242

Cc1cc(Nc2ncnc3nc(Nc4ccc(S(=O)(=O)NCCO)cc4)sc23)ccc1F

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EGFR P00533 19/20 0.57
CDK1 P06493 2/20 0.51
CCNB2 O95067 1/20 0.41
CCNE2 O96020 1/20 0.41
CDK4 P11802 1/20 0.41
CCNB1 P14635 1/20 0.41
CCND1 P24385 1/20 0.41
CCNE1 P24864 1/20 0.41
CDK2 P24941 1/20 0.41
CCND2 P30279 1/20 0.41
CCND3 P30281 1/20 0.41
CCNB3 Q8WWL7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13672635 0.90 EGFR (0.73) EGFRCDK1
SCHEMBL14461356 0.88 EGFR (0.56) EGFRCDK1CCNB2CCNE2CDK4
SCHEMBL13675235 0.85 EGFR (0.60) EGFRCDK1
SCHEMBL13675240 0.84 EGFR (0.79) EGFRCDK1
SCHEMBL13675047 0.83 EGFR (0.59) EGFRCDK1
SCHEMBL5069412 0.81 EGFR (0.57) EGFRCDK1
SCHEMBL13672628 0.81 EGFR (0.69) EGFRCDK1
SCHEMBL13675038 0.79 EGFR (0.83) EGFRCDK1
SCHEMBL13675052 0.77 EGFR (0.59) EGFRCDK1
SCHEMBL13675035 0.75 EGFR (0.81) EGFRCDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7605154-B2 ATP-protein kinase inhibitors; cytomegalovirus; contraceptive agents; cancer; N7-(3-ethynyl-phenyl)-N2-(4-piperidin-1-ylmethyl-phenyl)-thiazolo[4,5-d]pyrimidine-2,7-diamine JANSSEN PHARMACEUTICA N.V. (BE) 2009-10-20 US disclosed