SCHEMBL13680536

SCHEMBL13680536

Cc1cccc(-c2ccn3ccnc3c2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 2/20 0.53
TGFBR2 P37173 1/20 0.53
PIK3C3 Q8NEB9 1/20 0.44
ALDH1A1 P00352 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
GRM2 Q14416 1/20 0.40
PIK3CD O00329 1/20 0.40
ABL1 P00519 1/20 0.40
EGFR P00533 1/20 0.40
HCK P08631 1/20 0.40
SRC P12931 1/20 0.40
KDR P35968 1/20 0.40
PIK3CA P42336 1/20 0.40
PIK3CB P42338 1/20 0.40
MTOR P42345 1/20 0.40
PIK3CG P48736 1/20 0.40
EPHB4 P54760 1/20 0.40
PRKDC P78527 1/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5252715 0.82 KDR (0.50) PIK3C3PIK3CDABL1EGFRHCK
SCHEMBL13680666 0.81 TGFBR1 (0.68) TGFBR1TGFBR2PIK3CAFLT3HDAC6
SCHEMBL30186393 0.80 HSD17B2 (0.47) PIK3C3PIK3CACYP11B1CYP11B2
SCHEMBL14826051 0.80 PIK3C3 (0.51) TGFBR1TGFBR2PIK3C3PIK3CDABL1
SCHEMBL557143 0.80 SMN1; SMN2 (0.44) TGFBR1TGFBR2PIK3C3ALDH1A1L3MBTL1
Hydrochloric Acid SCHEMBL6544504 0.78 SMN1; SMN2 (0.43) TGFBR1TGFBR2PIK3C3ALDH1A1L3MBTL1
SCHEMBL3185826 0.78 PIK3C3 (0.45) TGFBR1TGFBR2PIK3C3PIK3CDABL1
SCHEMBL729192 0.77 KDR (0.52) PIK3C3ALDH1A1KDRCYP11B1CYP11B2
SCHEMBL3196822 0.76 TGFBR1 (0.54) TGFBR1TGFBR2PIK3C3PIK3CDABL1
SCHEMBL3325842 0.76 PIK3C3 (0.44) TGFBR1TGFBR2PIK3C3ALDH1A1PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed