SCHEMBL13680538

SCHEMBL13680538

COOSc1ccc(-c2nc(C)cs2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.43
CYP2E1 P05181 1/20 0.43
CYP2A6 P11509 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2B6 P20813 1/20 0.43
AOC3 Q16853 2/20 0.40
PDE10A Q9Y233 1/20 0.37
MAPT P10636 4/20 0.37
KDM4E B2RXH2 5/20 0.36
RAB9A P51151 4/20 0.36
NPC1 O15118 3/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
SREBF2 Q12772 1/20 0.36
ALDH1A1 P00352 4/20 0.36
POLB P06746 1/20 0.36
ATM Q13315 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
HPGD P15428 3/20 0.35
LMNA P02545 1/20 0.35
NFKB1 P19838 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680509 0.84 CYP3A4 (0.40) CYP3A4CYP2E1CYP2A6CYP2C9CYP2B6
SCHEMBL8198560 0.79 CYP3A4 (0.60) CYP3A4CYP2E1CYP2A6CYP2C9CYP2B6
SCHEMBL7905176 0.77 CYP3A4 (0.58) CYP3A4CYP2E1CYP2A6CYP2C9CYP2B6
SCHEMBL2096148 0.75 MAPT (0.61) AOC3MAPTKDM4ERAB9ANPC1
SCHEMBL13680944 0.74 KDM4E (0.41) MAPTKDM4ERAB9ANPC1SMN1; SMN2
SCHEMBL12180534 0.74 RAB9A (0.59) CYP3A4CYP2E1CYP2A6CYP2C9CYP2B6
SCHEMBL18725058 0.72 CYP3A4 (0.53) CYP3A4CYP2E1CYP2A6CYP2C9CYP2B6
SCHEMBL23367838 0.71 RAB9A (0.56) CYP3A4CYP2E1CYP2A6CYP2C9CYP2B6
SCHEMBL14438067 0.71 CYP3A4 (0.61) CYP3A4CYP2E1CYP2A6CYP2C9CYP2B6
SCHEMBL13680611 0.71 CYP3A4 (0.51) CYP3A4CYP2E1CYP2A6CYP2C9CYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed