SCHEMBL13680539

SCHEMBL13680539

COc1ccc(-c2nc(C)cs2)cn1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 4/20 0.61
CYP2A6 P11509 3/20 0.53
CYP2E1 P05181 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2B6 P20813 1/20 0.51
GRM5 P41594 1/20 0.44
CDC25A P30304 1/20 0.43
CDC25B P30305 1/20 0.43
PDGFRB P09619 1/20 0.43
PDGFRA P16234 1/20 0.43
PIK3CA P42336 2/20 0.43
PIK3CD O00329 1/20 0.43
PIP5K1C O60331 1/20 0.43
PIK3CB P42338 1/20 0.43
PI4KA P42356 1/20 0.43
PIK3CG P48736 1/20 0.43
PI4KB Q9UBF8 1/20 0.43
MKNK1 Q9BUB5 1/20 0.42
MKNK2 Q9HBH9 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680493 0.82 CYP2A6 (0.47) CYP19A1CYP2A6CYP2E1CYP3A4CYP2C9
SCHEMBL6840352 0.81 CYP3A4 (0.64) CYP19A1CYP2A6CYP2E1CYP3A4CYP2C9
SCHEMBL28731211 0.79 CYP19A1 (0.56) CYP19A1CYP2A6CDC25ACDC25BPDGFRB
SCHEMBL28731315 0.79 MAPT (0.65) CYP19A1CYP2A6CDC25ACDC25BPDGFRB
SCHEMBL18499144 0.79 NPSR1 (0.45) CYP19A1CYP2A6CYP2E1CYP3A4CYP2C9
SCHEMBL13680615 0.78 CYP2E1 (0.47) CYP19A1CYP2A6CYP2E1CYP3A4CYP2C9
SCHEMBL2141265 0.78 ALDH1A1 (0.61) CYP19A1CYP2A6MKNK1MKNK2CPT2
SCHEMBL27740381 0.77 CYP19A1 (0.56) CYP19A1CYP2A6MKNK1MKNK2CPT2
SCHEMBL2925411 0.77 CYP19A1 (0.56) CYP19A1CYP2A6PIK3CGMKNK1MKNK2
SCHEMBL13680530 0.77 CYP2A6 (0.54) CYP2A6CYP2E1CYP3A4CYP2C9CYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed