SCHEMBL13680530

SCHEMBL13680530

Cc1csc(-c2ccc(F)nc2)n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 4/20 0.54
CYP2B6 P20813 4/20 0.54
CYP3A4 P08684 4/20 0.54
CYP2E1 P05181 2/20 0.54
CYP2C9 P11712 1/20 0.54
CYP2C19 P33261 2/20 0.50
PDE10A Q9Y233 1/20 0.44
AOC3 Q16853 2/20 0.43
GRM5 P41594 1/20 0.42
NTMT1 Q9BV86 1/20 0.40
MAPT P10636 1/20 0.39
GABRA1 P14867 1/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
GABRA5 P31644 1/20 0.38
GABRA3 P34903 1/20 0.38
GABRA2 P47869 1/20 0.38
TLR9 Q9NR96 1/20 0.37
TLR8 Q9NR97 1/20 0.37
TLR7 Q9NYK1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6840352 0.84 CYP3A4 (0.64) CYP2A6CYP2B6CYP3A4CYP2E1CYP2C9
SCHEMBL8198560 0.79 CYP3A4 (0.60) CYP2A6CYP2B6CYP3A4CYP2E1CYP2C9
SCHEMBL13680533 0.79 CYP2E1 (0.50) CYP2A6CYP2B6CYP3A4CYP2E1CYP2C9
SCHEMBL2092693 0.78 KDM4E (0.56) CYP2A6CYP2B6CYP3A4CYP2E1CYP2C9
SCHEMBL7905176 0.77 CYP3A4 (0.58) CYP2A6CYP2B6CYP3A4CYP2E1CYP2C9
SCHEMBL13680575 0.77 CYP2E1 (0.51) CYP2A6CYP2B6CYP3A4CYP2E1CYP2C9
SCHEMBL13680539 0.77 CYP19A1 (0.61) CYP2A6CYP2B6CYP3A4CYP2E1CYP2C9
SCHEMBL13680744 0.76 CYP3A4 (0.53) CYP2A6CYP2B6CYP3A4CYP2E1CYP2C9
SCHEMBL13681280 0.76 CYP2E1 (0.50) CYP2A6CYP2B6CYP3A4CYP2E1CYP2C9
SCHEMBL16603176 0.76 LMNA (0.46) CYP2A6CYP2B6CYP3A4CYP2E1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed