SCHEMBL13680625

SCHEMBL13680625

Cc1csc(-c2ccc3[nH]c(=O)[nH]c3c2)n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC25A P30304 1/20 0.56
CDC25B P30305 1/20 0.56
CDC25C P30307 1/20 0.56
DUSP3 P51452 1/20 0.56
PDE3B Q13370 2/20 0.53
PDE3A Q14432 2/20 0.53
GRIA1 P42261 5/20 0.50
CACNG8 Q8WXS5 5/20 0.50
TLR9 Q9NR96 1/20 0.48
TLR8 Q9NR97 1/20 0.48
TLR7 Q9NYK1 1/20 0.48
GABRA1 P14867 3/20 0.43
GABRG2 P18507 3/20 0.43
GABRB3 P28472 3/20 0.43
GABRA5 P31644 3/20 0.43
GABRA3 P34903 3/20 0.43
GABRA2 P47869 3/20 0.43
CYP2E1 P05181 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2A6 P11509 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680627 0.81 CA12 (0.51) CDC25ACDC25BCDC25CDUSP3PDE3B
SCHEMBL13680622 0.79 PDE3B (0.56) CDC25ACDC25BCDC25CDUSP3PDE3B
SCHEMBL13680624 0.77 NPC1 (0.51) TLR9TLR8TLR7CYP2E1CYP3A4
SCHEMBL19626747 0.77 CDC25A (0.58) CDC25ACDC25BCDC25CDUSP3PDE3B
SCHEMBL6200129 0.76 CDC25A (0.64) CDC25ACDC25BCDC25CDUSP3
SCHEMBL13680995 0.76 CDC25A (0.48) CDC25ACDC25BCDC25CDUSP3PDE3B
SCHEMBL8198560 0.75 CYP3A4 (0.60) TLR9TLR8TLR7GABRA1GABRG2
SCHEMBL13680616 0.75 EGFR (0.51) TLR9TLR8TLR7CYP2E1CYP3A4
SCHEMBL13680617 0.74 GSK3B (0.61) TLR9TLR8TLR7CYP2E1CYP3A4
SCHEMBL19625362 0.74 CDC25A (0.55) CDC25ACDC25BCDC25CDUSP3PDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed