SCHEMBL13680642

SCHEMBL13680642

Cc1cccc(-c2ccc3c(c2)CCC3=O)c1

nearest known ligand 0.64

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 5/20 0.64
PARP11 Q9NR21 5/20 0.64
CYP1A2 P05177 1/20 0.59
CYP11B1 P15538 1/20 0.59
CYP11B2 P19099 1/20 0.59
HSD17B1 P14061 5/20 0.58
PGR P06401 2/20 0.54
FYN P06241 1/20 0.51
CLK4 Q9HAZ1 1/20 0.51
DYRK1B Q9Y463 1/20 0.51
CASP1 P29466 1/20 0.47
CASP7 P55210 1/20 0.47
HSD17B10 Q99714 1/20 0.47
GRM5 P41594 1/20 0.44
GRM1 Q13255 1/20 0.43
DHODH Q02127 1/20 0.42
MAPK14 Q16539 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4424565 0.90 PARP10 (0.61) PARP10PARP11CYP1A2CYP11B1CYP11B2
SCHEMBL19100757 0.86 HSD17B1 (0.62) PARP10PARP11CYP1A2CYP11B1CYP11B2
SCHEMBL1747435 0.84 HSD17B1 (0.69) PARP10PARP11CYP1A2CYP11B1CYP11B2
SCHEMBL28655414 0.84 HSD17B1 (0.78) PARP10PARP11CYP1A2CYP11B1CYP11B2
SCHEMBL1745161 0.82 HSD17B1 (0.71) PARP10PARP11CYP1A2CYP11B1CYP11B2
SCHEMBL3630871 0.80 HSD17B1 (0.54) PARP10PARP11CYP1A2CYP11B1CYP11B2
Dimethylamine SCHEMBL3994802 0.80 HSD17B1 (0.63) PARP10PARP11CYP1A2CYP11B1CYP11B2
SCHEMBL3989386 0.80 CASP1 (0.66) PARP10PARP11CYP1A2CYP11B1CYP11B2
SCHEMBL6192593 0.80 PARP10 (0.64) PARP10PARP11CYP1A2CYP11B1CYP11B2
SCHEMBL29726014 0.80 CASP1 (0.59) PARP10PARP11CYP1A2CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed