SCHEMBL13680669

SCHEMBL13680669

CNC(=S)c1ccc(-c2cccc(C)n2)cn1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.49
CYP2A6 P11509 1/20 0.46
MAPT P10636 2/20 0.44
TGFBR1 P36897 10/20 0.43
CCR1 P32246 1/20 0.43
CCR8 P51685 1/20 0.43
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
MAPK14 Q16539 1/20 0.38
SIK2 Q9H0K1 1/20 0.38
PAK1 Q13153 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13681313 0.78 CYP2A6 (0.45) GRM5CYP2A6TGFBR1CCR1CCR8
SCHEMBL13680554 0.78 GRM5 (0.53) GRM5CYP2A6TGFBR1CCR1CCR8
SCHEMBL30146674 0.76 CYP2A6 (0.65) GRM5CYP2A6TGFBR1CCR1CCR8
SCHEMBL3421947 0.76 CYP2A6 (0.65) GRM5CYP2A6TGFBR1CCR1CCR8
SCHEMBL13051887 0.73 CCR1 (0.59) GRM5CYP2A6TGFBR1CCR1CCR8
SCHEMBL24673834 0.71 CYP2A6 (0.54) GRM5CYP2A6TGFBR1CCR1CCR8
SCHEMBL29457509 0.71 CYP2A6 (0.54) GRM5CYP2A6TGFBR1CCR1CCR8
SCHEMBL16835922 0.71 CYP2A6 (0.54) GRM5CYP2A6TGFBR1CCR1CCR8
SCHEMBL1743453 0.71 CYP2A6 (0.54) GRM5CYP2A6TGFBR1CCR1CCR8
SCHEMBL13680479 0.71 CYP2A6 (0.54) GRM5CYP2A6MAPTTGFBR1CCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed