SCHEMBL13680677

SCHEMBL13680677

CSc1ncc(-c2cccc(C)n2)cn1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.54
CCR8 P51685 1/20 0.54
CYP2A6 P11509 1/20 0.51
METAP2 P50579 1/20 0.43
TGFBR1 P36897 10/20 0.41
SCN9A Q15858 1/20 0.39
MAPK14 Q16539 1/20 0.38
GRM5 P41594 1/20 0.38
NOS3 P29474 1/20 0.36
NOS2 P35228 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
BRS3 P32247 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680679 0.82 CCR1 (0.60) CCR1CCR8CYP2A6METAP2TGFBR1
SCHEMBL23243808 0.82 SCN9A (0.37) CCR1CCR8CYP2A6SCN9AMEN1
SCHEMBL13680673 0.79 CCR1 (0.56) CCR1CCR8CYP2A6METAP2TGFBR1
SCHEMBL13681326 0.79 CCR1 (0.50) CCR1CCR8CYP2A6METAP2TGFBR1
SCHEMBL16068071 0.78 SCN9A (0.45) TGFBR1SCN9A
SCHEMBL30146674 0.77 CYP2A6 (0.65) CCR1CCR8CYP2A6METAP2TGFBR1
SCHEMBL3421947 0.77 CYP2A6 (0.65) CCR1CCR8CYP2A6METAP2TGFBR1
SCHEMBL13680586 0.76 CCR1 (0.52) CCR1CCR8CYP2A6METAP2TGFBR1
SCHEMBL13680674 0.76 CCR1 (0.52) CCR1CCR8CYP2A6METAP2TGFBR1
SCHEMBL13680680 0.76 CYP2A6 (0.54) CCR1CCR8CYP2A6METAP2TGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed