SCHEMBL13680683

SCHEMBL13680683

Cc1cccc(-c2cnc(=O)[nH]c2)n1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.50
CCR1 P32246 1/20 0.47
CCR8 P51685 1/20 0.47
METAP2 P50579 2/20 0.42
LYN P07948 1/20 0.42
TGFBR1 P36897 9/20 0.40
SIK2 Q9H0K1 2/20 0.40
MAPK14 Q16539 1/20 0.38
GRM5 P41594 1/20 0.37
STK4 Q13043 1/20 0.36
STK3 Q13188 1/20 0.36
STK26 Q9P289 1/20 0.36
STK24 Q9Y6E0 1/20 0.36
BRS3 P32247 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680690 0.77 CCR1 (0.50) CYP2A6CCR1CCR8METAP2TGFBR1
SCHEMBL15326994 0.76 CCR1 (0.54) CYP2A6CCR1CCR8METAP2TGFBR1
SCHEMBL29590240 0.76 CCR1 (0.54) CYP2A6CCR1CCR8METAP2TGFBR1
SCHEMBL30146674 0.75 CYP2A6 (0.65) CYP2A6CCR1CCR8METAP2TGFBR1
SCHEMBL3421947 0.75 CYP2A6 (0.65) CYP2A6CCR1CCR8METAP2TGFBR1
SCHEMBL13680655 0.75 LYN (0.57) METAP2LYN
SCHEMBL1743453 0.75 CYP2A6 (0.54) CYP2A6CCR1CCR8METAP2TGFBR1
SCHEMBL12863970 0.74 LYN (0.44) METAP2LYN
SCHEMBL2352218 0.73 AKT1 (0.52) LYNSTK3
SCHEMBL13680679 0.73 CCR1 (0.60) CYP2A6CCR1CCR8METAP2TGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed