SCHEMBL13680690

SCHEMBL13680690

Cc1cccc(-c2ccc(=O)[nH]c2)n1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.50
CCR8 P51685 1/20 0.50
CYP2A6 P11509 1/20 0.49
MAPT P10636 2/20 0.47
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
THRB P10828 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
TGFBR1 P36897 6/20 0.42
METAP2 P50579 2/20 0.41
MAPK14 Q16539 1/20 0.39
SIK2 Q9H0K1 1/20 0.39
ATR Q13535 2/20 0.38
PDGFRB P09619 1/20 0.38
PDGFRA P16234 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10999711 0.78 CYP11B1 (0.46) MAPTKDM4EALDH1A1THRBL3MBTL1
SCHEMBL11448878 0.78 MEN1 (0.48) MAPTKDM4EALDH1A1THRBL3MBTL1
SCHEMBL13680683 0.77 CYP2A6 (0.50) CCR1CCR8CYP2A6TGFBR1METAP2
SCHEMBL3422361 0.77 CCR1 (0.75) CCR1CCR8CYP2A6MAPTALDH1A1
SCHEMBL13680450 0.76 CA12 (0.53) CCR1CCR8CYP2A6MAPTTHRB
SCHEMBL27973522 0.76 CCR1 (0.50) CCR1CCR8CYP2A6MAPTTGFBR1
SCHEMBL10999876 0.75 KDM4E (0.48) MAPTKDM4EALDH1A1THRBL3MBTL1
SCHEMBL10999258 0.75 MEN1 (0.44) MAPTKDM4EALDH1A1THRBL3MBTL1
SCHEMBL10997580 0.74 ALDH1A1 (0.41) MAPTKDM4EALDH1A1THRBL3MBTL1
SCHEMBL13680558 0.73 GRIA1 (0.59) CCR1CCR8CYP2A6TGFBR1METAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed