SCHEMBL13680697

SCHEMBL13680697

CNc1ncc(-c2cccc(C)n2)s1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 7/20 0.51
CCR1 P32246 1/20 0.47
CCR8 P51685 1/20 0.47
CCNT1 O60563 3/20 0.46
CCNA2 P20248 3/20 0.46
CDK2 P24941 3/20 0.46
CDK9 P50750 3/20 0.46
CDK1 P06493 2/20 0.46
CCNB1 P14635 2/20 0.46
CDK7 P50613 2/20 0.46
CCNH P51946 2/20 0.46
CCNA1 P78396 2/20 0.46
MAPK14 Q16539 2/20 0.41
LMNA P02545 1/20 0.41
CYP2A6 P11509 1/20 0.39
METAP2 P50579 1/20 0.39
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15859041 0.80 CCR1 (0.54) KDRCCR1CCR8MAPK14CYP2A6
SCHEMBL13680693 0.77 CCR1 (0.50) KDRCCR1CCR8MAPK14CYP2A6
SCHEMBL2865766 0.75 KDR (0.59) KDRCCNT1CCNA2CDK2CDK9
SCHEMBL6169965 0.75 KDR (0.46) KDRCCR1CCR8CDK7MAPK14
SCHEMBL6169974 0.75 KDR (0.46) KDRCCR1CCR8CCNT1CCNA2
SCHEMBL13680698 0.74 CCR1 (0.47) KDRCCR1CCR8MAPK14CYP2A6
SCHEMBL13680692 0.74 DYRK1A (0.56) KDRCCR1CCR8MAPK14CYP2A6
SCHEMBL13513650 0.74 KDR (0.66) KDRCDK2LMNANPC1RAB9A
SCHEMBL6169672 0.73 KDR (0.44) KDRCCNT1CCNA2CDK2CDK9
SCHEMBL12715402 0.73 CDK2 (0.51) CCNT1CCNA2CDK2CDK9CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed