SCHEMBL13680693

SCHEMBL13680693

Cc1cccc(-c2cnc(N)s2)n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.50
CCR8 P51685 1/20 0.50
BACE1 P56817 1/20 0.47
NOS3 P29474 1/20 0.47
NOS2 P35228 1/20 0.47
MAPK14 Q16539 3/20 0.44
TGFBR1 P36897 6/20 0.43
NOS1 P29475 1/20 0.42
NPC1 O15118 3/20 0.42
MAPT P10636 3/20 0.42
RAB9A P51151 3/20 0.42
ALDH1A1 P00352 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
CSNK2A1 P68400 1/20 0.41
CYP2A6 P11509 1/20 0.41
METAP2 P50579 1/20 0.41
KDR P35968 1/20 0.40
KDM4E B2RXH2 1/20 0.38
TP53 P04637 1/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15859041 0.82 CCR1 (0.54) CCR1CCR8NOS3NOS2MAPK14
SCHEMBL13681316 0.79 LOXL2 (0.50) CCR1CCR8NOS3NOS2TGFBR1
SCHEMBL13680692 0.77 DYRK1A (0.56) CCR1CCR8NOS3NOS2MAPK14
SCHEMBL13680697 0.77 KDR (0.51) CCR1CCR8NOS3NOS2MAPK14
SCHEMBL13680698 0.77 CCR1 (0.47) CCR1CCR8NOS3NOS2MAPK14
SCHEMBL13629651 0.74 ASIC3 (0.48) BACE1NOS3NOS2NOS1MAPT
SCHEMBL14606354 0.74 CCR1 (0.62) CCR1CCR8NOS3NOS2MAPK14
SCHEMBL17889606 0.73 MAPK14 (0.61) CCR1CCR8NOS3NOS2MAPK14
SCHEMBL31093398 0.72 LMNA (0.48) BACE1MAPK14NOS1NPC1MAPT
SCHEMBL12775047 0.71 NOS3 (0.74) CCR1CCR8NOS3NOS2TGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed