SCHEMBL13680756

SCHEMBL13680756

Cc1csc(-c2cnc(N(C)C)cn2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.46
ADORA2A P29274 3/20 0.39
ADORA1 P30542 3/20 0.39
CYP3A4 P08684 2/20 0.38
CYP2E1 P05181 1/20 0.38
CYP2A6 P11509 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2B6 P20813 1/20 0.38
SRC P12931 1/20 0.37
CDK2 P24941 1/20 0.37
ZAP70 P43403 1/20 0.37
SYK P43405 1/20 0.37
NOS1 P29475 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TP53 P04637 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680575 0.75 CYP2E1 (0.51) PDE10AADORA2AADORA1CYP3A4CYP2E1
SCHEMBL13681060 0.74 NPC1 (0.31) SMN1; SMN2
SCHEMBL13680745 0.73 PDE10A (0.46) PDE10AADORA2AADORA1CYP3A4CYP2E1
SCHEMBL13680739 0.70 ADORA2A (0.49) PDE10AADORA2AADORA1CYP3A4CYP2E1
SCHEMBL5912824 0.70 PDE10A (0.59) PDE10ACYP3A4CYP2E1CYP2A6CYP2C9
SCHEMBL18157874 0.69 SMN1; SMN2 (0.55) PDE10AADORA2AADORA1CYP3A4CYP2E1
SCHEMBL13680687 0.68 CCR1 (0.55) ADORA2AADORA1CYP3A4CYP2A6CKS1B
SCHEMBL46324 0.67 MEN1 (0.37) CYP3A4CYP2A6MEN1KMT2AALDH1A1
SCHEMBL13680737 0.67 ADORA2A (0.39) PDE10AADORA2AADORA1CYP3A4CYP2E1
SCHEMBL19396093 0.66 PDE10A (0.39) PDE10ACYP3A4CYP2E1CYP2A6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed