SCHEMBL13680575

SCHEMBL13680575

Cc1csc(-c2ccc(N(C)C)nc2)n1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2E1 P05181 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2A6 P11509 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2B6 P20813 1/20 0.51
APP P05067 6/20 0.45
PDE10A Q9Y233 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA1 P30542 1/20 0.41
AOC3 Q16853 3/20 0.39
PRMT1 Q99873 3/20 0.38
MAPT P10636 1/20 0.38
MAP3K11 Q16584 1/20 0.38
CRHR1 P34998 2/20 0.37
TLR8 Q9NR97 1/20 0.37
TLR7 Q9NYK1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6840352 0.81 CYP3A4 (0.64) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL13680739 0.80 ADORA2A (0.49) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL13680530 0.77 CYP2A6 (0.54) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL8198560 0.76 CYP3A4 (0.60) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL13680756 0.75 PDE10A (0.46) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL13680954 0.75 KDM4E (0.40) APPPRMT1MAPT
SCHEMBL7905176 0.74 CYP3A4 (0.58) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL13680539 0.74 CYP19A1 (0.61) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL23158936 0.73 APP (0.47) APPADORA2AADORA1AOC3MAPT
SCHEMBL13680744 0.73 CYP3A4 (0.53) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed