SCHEMBL13680745

SCHEMBL13680745

Cc1csc(-c2ccc(N(C)C)nn2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.46
TP53 P04637 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
NPC1 O15118 1/20 0.46
USP2 O75604 1/20 0.46
PKM P14618 1/20 0.46
RAB9A P51151 1/20 0.46
ADORA2A P29274 3/20 0.42
ADORA1 P30542 2/20 0.42
CYP3A4 P08684 2/20 0.38
CYP2E1 P05181 1/20 0.38
CYP2A6 P11509 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2B6 P20813 1/20 0.38
SRC P12931 1/20 0.37
CDK2 P24941 1/20 0.37
ZAP70 P43403 1/20 0.37
SYK P43405 1/20 0.37
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680756 0.73 PDE10A (0.46) PDE10ATP53SMN1; SMN2ADORA2AADORA1
SCHEMBL13681053 0.73 RAB9A (0.37) TP53SMN1; SMN2NPC1USP2PKM
SCHEMBL13680575 0.72 CYP2E1 (0.51) PDE10AADORA2AADORA1CYP3A4CYP2E1
SCHEMBL10842162 0.70 NPC1 (0.59) TP53SMN1; SMN2NPC1USP2PKM
SCHEMBL13680688 0.69 CCR1 (0.57) TP53SMN1; SMN2NPC1USP2PKM
SCHEMBL13377800 0.69 PDE10A (0.67) PDE10ATP53SMN1; SMN2RAB9AADORA2A
SCHEMBL18157874 0.69 SMN1; SMN2 (0.55) PDE10ATP53SMN1; SMN2NPC1RAB9A
SCHEMBL4278637 0.68 NPC1 (0.58) TP53SMN1; SMN2NPC1USP2PKM
SCHEMBL2629425 0.67 RAB9A (0.48) TP53SMN1; SMN2NPC1USP2PKM
SCHEMBL10842285 0.66 SMN1; SMN2 (0.69) TP53SMN1; SMN2NPC1USP2PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed