SCHEMBL13683032

SCHEMBL13683032

CC(C)n1nc(CN2CCOCC2)c(Cl)c1-c1ccccn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
CYP2A13 Q16696 3/20 0.39
TGFBR1 P36897 2/20 0.39
MAPK13 O15264 1/20 0.39
MAPK12 P53778 1/20 0.39
MAPK11 Q15759 1/20 0.39
MAPK14 Q16539 1/20 0.39
PIK3CA P42336 1/20 0.38
MTOR P42345 1/20 0.38
KMT2A Q03164 2/20 0.38
ALDH1A1 P00352 2/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KDM4E B2RXH2 1/20 0.37
GLA P06280 1/20 0.37
GAA P10253 1/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13184392 0.86 CYP2A13 (0.40) SLC2A1NPSR1CYP2A13KMT2AALDH1A1
SCHEMBL16200163 0.85 SLC2A1 (0.46) SLC2A1NPSR1CYP2A13TGFBR1MAPK13
SCHEMBL16200193 0.83 SLC2A1 (0.42) SLC2A1NPSR1CYP2A13TGFBR1MAPK13
SCHEMBL14044135 0.80 SLC2A1 (0.48) SLC2A1NPSR1CYP2A13TGFBR1PIK3CA
SCHEMBL13683095 0.78 CA1 (0.38) LMNAKDM4E
SCHEMBL14044138 0.78 ADORA2A (0.40) NPSR1CYP2A13HTTSMN1; SMN2KCNH2
SCHEMBL14044093 0.76 METAP1 (0.36) KMT2AMEN1LMNAKDM4EMETAP2
SCHEMBL13683031 0.76 ADORA1 (0.36) KMT2AMEN1LMNAKDM4EMETAP2
SCHEMBL16200157 0.72 CYP2A13 (0.43) SLC2A1NPSR1CYP2A13MAPK13MAPK12
SCHEMBL16200392 0.68 SLC2A1 (0.47) SLC2A1NPSR1CYP2A13TGFBR1MAPK13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8324216-B2 Substituted piperazines CHEMOCENTRYX, INC. (US) 2012-12-04 US disclosed
US-7589199-B2 Substituted piperazines CHEMOCENTRYX, INC. (US) 2009-09-15 US disclosed
US-7435831-B2 Bicyclic and bridged nitrogen heterocycles CHEMOCENTRYX, INC. (US) 2008-10-14 US disclosed