SCHEMBL14044138

SCHEMBL14044138

CC(C)n1nc(CN2CCOCC2)c(Cl)c1-c1nccs1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.40
ADORA1 P30542 1/20 0.40
KCNH2 Q12809 8/20 0.39
SMN1; SMN2 Q16637 2/20 0.36
CYP2A13 Q16696 2/20 0.34
HTT P42858 1/20 0.34
HRH3 Q9Y5N1 3/20 0.33
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13184392 0.81 CYP2A13 (0.40) CYP2A13HRH3NPSR1
SCHEMBL14044109 0.80 ADORA2A (0.40) ADORA2AADORA1KCNH2SMN1; SMN2CYP2A13
SCHEMBL13683032 0.78 SLC2A1 (0.42) KCNH2SMN1; SMN2CYP2A13HTTNPSR1
SCHEMBL16200394 0.71 ADORA2A (0.42) ADORA2AADORA1KCNH2SMN1; SMN2CYP2A13
SCHEMBL27721308 0.69 HRH3 (0.63) ADORA2AADORA1SMN1; SMN2HTTHRH3
SCHEMBL16200157 0.68 CYP2A13 (0.43) CYP2A13HRH3NPSR1
SCHEMBL5200192 0.65 SMN1; SMN2 (0.37) KCNH2SMN1; SMN2CYP2A13HRH3
SCHEMBL952226 0.65 ALOX15 (0.55) ADORA2AADORA1SMN1; SMN2HTT
SCHEMBL16200163 0.64 SLC2A1 (0.46) CYP2A13NPSR1
SCHEMBL16200193 0.63 SLC2A1 (0.42) CYP2A13NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7435830-B2 Bicyclic and bridged nitrogen heterocycles CHEMOCENTRYX, INC. (US) 2008-10-14 US disclosed