SCHEMBL13683095

SCHEMBL13683095

CC(C)n1nc(CO)c(Cl)c1-c1ccccn1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA4 P22748 1/20 0.38
CA9 Q16790 1/20 0.38
ADORA1 P30542 1/20 0.38
RET P07949 5/20 0.36
TRPM8 Q7Z2W7 1/20 0.34
METAP1 P53582 2/20 0.34
KLKB1 P03952 2/20 0.34
POLB P06746 2/20 0.34
CCR1 P32246 2/20 0.34
CCR5 P51681 2/20 0.34
CCR8 P51685 2/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
CYP1A2 P05177 1/20 0.34
BLM P54132 1/20 0.34
HIF1A Q16665 1/20 0.34
DOHH Q9BU89 1/20 0.34
P4HTM Q9NXG6 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14044093 0.84 METAP1 (0.36) ADORA1RETMETAP1POLBCCR1
SCHEMBL13683031 0.84 ADORA1 (0.36) ADORA1RETMETAP1KLKB1POLB
SCHEMBL14044137 0.83 ALDH1A1 (0.32) POLBMPO
SCHEMBL16200177 0.82 CA1 (0.43) CA1CA2CA4CA9METAP1
SCHEMBL13683032 0.78 SLC2A1 (0.42) KDM4ELMNA
SCHEMBL13683059 0.69 ADORA1 (0.40) ADORA1RETMETAP1KLKB1POLB
SCHEMBL16200192 0.66 IDO1 (0.36)
SCHEMBL16200168 0.66 METAP1 (0.38) METAP1POLBCCR1CCR5CCR8
SCHEMBL15048580 0.65 KDM4E (0.45) ADORA1RETMETAP1POLBCCR1
SCHEMBL16200366 0.65 METAP1 (0.44) METAP1POLBCCR1CCR5CCR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720545-B1 BICYCLIC AND BRIDGED NITROGEN HETEROCYCLES CHEMOCENTRYX INC (US) 2014-10-29 EP disclosed
US-7589199-B2 Substituted piperazines CHEMOCENTRYX, INC. (US) 2009-09-15 US disclosed
US-7435830-B2 Bicyclic and bridged nitrogen heterocycles CHEMOCENTRYX, INC. (US) 2008-10-14 US disclosed