SCHEMBL13683178

SCHEMBL13683178

Cc1nn(C)c(C(=O)c2ccccn2)c1F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.45
ALDH1A1 P00352 1/20 0.44
HSD17B14 Q9BPX1 1/20 0.43
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
L3MBTL1 Q9Y468 3/20 0.41
LMNA P02545 1/20 0.41
NAPRT Q6XQN6 1/20 0.41
P4HTM Q9NXG6 1/20 0.41
KDM4E B2RXH2 2/20 0.39
GRM4 Q14833 1/20 0.38
CTNNB1 P35222 2/20 0.38
WNT3A P56704 2/20 0.38
RAB9A P51151 3/20 0.37
GSK3B P49841 1/20 0.37
NPC1 O15118 2/20 0.37
GLA P06280 1/20 0.37
AGTR1 P30556 1/20 0.36
RIPK1 Q13546 1/20 0.36
TLR7 Q9NYK1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16200362 0.80 KMT2A (0.42) KMT2AALDH1A1CES2CES1L3MBTL1
SCHEMBL13683133 0.77 KMT2A (0.45) KMT2AALDH1A1HSD17B14CES2CES1
SCHEMBL6919650 0.75 KMT2A (0.46) KMT2AALDH1A1HSD17B14CES2CES1
SCHEMBL9197914 0.75 TP53 (0.49) ALDH1A1L3MBTL1LMNARAB9ANPC1
SCHEMBL13184261 0.72 BAZ2B (0.49) KMT2AALDH1A1HSD17B14CES2CES1
SCHEMBL31369148 0.70 KMT2A (0.75) KMT2AALDH1A1HSD17B14CES2CES1
SCHEMBL87791 0.70 KMT2A (0.75) KMT2AALDH1A1HSD17B14CES2CES1
SCHEMBL13184427 0.70 KMT2A (0.46) KMT2AALDH1A1HSD17B14CES2CES1
SCHEMBL13683180 0.69 KDM4E (0.41) KMT2AALDH1A1L3MBTL1LMNAKDM4E
SCHEMBL19556155 0.69 L3MBTL1 (0.42) KMT2AALDH1A1L3MBTL1LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7589199-B2 Substituted piperazines CHEMOCENTRYX, INC. (US) 2009-09-15 US disclosed