SCHEMBL13700178

SCHEMBL13700178

CN(CCO)Cc1cccc(C(=O)Nc2c(C(N)=O)oc3c(F)cc(F)cc23)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK10 P53779 4/20 0.40
HSD17B10 Q99714 3/20 0.40
TSHR P16473 2/20 0.40
HPGD P15428 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TP53 P04637 4/20 0.40
MAPT P10636 3/20 0.40
AHR P35869 1/20 0.40
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 2/20 0.38
HASPIN Q8TF76 1/20 0.36
CHEK1 O14757 1/20 0.36
SIGMAR1 Q99720 5/20 0.36
TMEM97 Q5BJF2 4/20 0.36
ACKR3 P25106 3/20 0.35
ROCK2 O75116 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13700141 0.91 TSHR (0.43) MAPK10HSD17B10TSHRHPGDMEN1
SCHEMBL13700196 0.91 MAPK10 (0.41) MAPK10HSD17B10TSHRHPGDMEN1
SCHEMBL13700207 0.89 MAPK10 (0.39) MAPK10HSD17B10TSHRHPGDMEN1
SCHEMBL13700156 0.86 CYP2D6 (0.44) MAPK10HSD17B10TSHRHPGDMEN1
SCHEMBL13700349 0.86 MAPK10 (0.35) MAPK10HSD17B10TSHRHPGDMEN1
SCHEMBL13700163 0.85 MAPK10 (0.44) MAPK10HSD17B10TSHRHPGDMEN1
SCHEMBL13700162 0.84 TSHR (0.36) MAPK10HSD17B10TSHRHPGDMEN1
SCHEMBL13700241 0.84 PTGDR2 (0.36) MAPK10HSD17B10TSHRHPGDMEN1
SCHEMBL13699897 0.83 MAPK10 (0.45) MAPK10HSD17B10TSHRHPGDMEN1
SCHEMBL13700197 0.82 CHRM3 (0.43) MAPK10HSD17B10TSHRHPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090239860-A1 NOVEL BENZOFURAN DERIVATIVE, MEDICINAL COMPOSITION CONTAINING THE SAME, AND USES OF THESE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-09-24 US disclosed
US-20090239860-A1 NOVEL BENZOFURAN DERIVATIVE, MEDICINAL COMPOSITION CONTAINING THE SAME, AND USES OF THESE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-09-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090239860-A1 NOVEL BENZOFURAN DERIVATIVE, MEDICINAL COMPOSITION CONTAINING THE SAME, AND USES OF THESE ADORA2A, ADORA2B, HTR1F MAPK10 3802/4885HSD17B10 1250/4885TSHR 231/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.