SCHEMBL13705609

SCHEMBL13705609

Nc1ccc(F)c(C(=O)Nc2cnc3[nH]cc(-c4cccc(CN5CCOCC5)c4)c3c2)c1F

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 3/20 0.54
GSK3B P49841 3/20 0.54
PRKD3 O94806 3/20 0.54
MAP4K4 O95819 3/20 0.54
EGFR P00533 3/20 0.54
NTRK1 P04629 3/20 0.54
LCK P06239 3/20 0.54
FYN P06241 3/20 0.54
AXL P30530 3/20 0.54
FLT4 P35916 3/20 0.54
FLT3 P36888 3/20 0.54
FRK P42685 3/20 0.54
CLK2 P49760 3/20 0.54
MAP4K2 Q12851 3/20 0.54
CAMK2B Q13554 3/20 0.54
CAMK2G Q13555 3/20 0.54
CAMK2D Q13557 3/20 0.54
PTK6 Q13882 3/20 0.54
NTRK3 Q16288 3/20 0.54
PKN2 Q16513 3/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13705558 0.87 PRKD3 (0.56) CDK1GSK3BPRKD3MAP4K4EGFR
SCHEMBL1773762 0.85 BRAF (0.63)
SCHEMBL13705611 0.83 BTK (0.59) CDK1GSK3BPRKD3MAP4K4EGFR
SCHEMBL2356446 0.81 CYP2C19 (0.52) EGFRPTK6MAP4K5KDRMAP3K20
SCHEMBL14235967 0.79 BRAF (0.45) CLK2DYRK1ACDK5
SCHEMBL13705600 0.79 PRKD3 (0.63) CDK1GSK3BPRKD3MAP4K4EGFR
SCHEMBL13705608 0.79 DYRK1A (0.68) CDK1GSK3BPRKD3MAP4K4EGFR
SCHEMBL13705602 0.79 BTK (0.62) CDK1GSK3BPRKD3MAP4K4EGFR
SCHEMBL13705610 0.79 ALK (0.57) CDK1GSK3BPRKD3MAP4K4EGFR
SCHEMBL13705612 0.77 CLK4 (0.64) CDK1GSK3BPRKD3MAP4K4EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009111278-A2 RAF INHIBITOR COMPOUNDS AND METHODS OF USE THEREOF ARRAY BIOPHARMA INC. (US) 2009-09-11 WO disclosed