SCHEMBL13708282

SCHEMBL13708282

CCOC(=O)c1coc(C(=O)c2sc(NC(=O)c3ccccc3C)c(C#N)c2N)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 4/20 0.61
ALDH1A1 P00352 8/20 0.49
HPGD P15428 6/20 0.49
MAPT P10636 7/20 0.46
MEN1 O00255 5/20 0.46
KMT2A Q03164 5/20 0.46
SMN1; SMN2 Q16637 5/20 0.46
RAB9A P51151 4/20 0.46
HTT P42858 4/20 0.46
POLB P06746 3/20 0.46
LMNA P02545 3/20 0.46
MAPK1 P28482 2/20 0.46
KDM4E B2RXH2 1/20 0.46
MELK Q14680 1/20 0.44
CRHBP P24387 1/20 0.44
CRHR2 Q13324 1/20 0.44
PKM P14618 1/20 0.44
GAA P10253 2/20 0.44
NPC1 O15118 1/20 0.44
TP53 P04637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4477192 0.76 BRAF (0.54) BRAFALDH1A1MAPTMEN1KMT2A
SCHEMBL13708307 0.69 MELK (0.54) ALDH1A1HPGDMAPTMEN1KMT2A
SCHEMBL4489057 0.66 MELK (0.45) BRAFALDH1A1HPGDMEN1KMT2A
SCHEMBL4478646 0.65 CFTR (0.51) BRAFALDH1A1HPGDMAPTMEN1
SCHEMBL5232976 0.63 SMN1; SMN2 (1.00) ALDH1A1HPGDMAPTMEN1KMT2A
SCHEMBL3419606 0.63 MEN1 (0.64) BRAFALDH1A1HPGDMAPTMEN1
SCHEMBL15183729 0.63 RAB9A (1.00) ALDH1A1HPGDMAPTMEN1KMT2A
SCHEMBL3016097 0.62 CA12 (0.52) ALDH1A1HPGDMAPTMEN1KMT2A
SCHEMBL3279549 0.62 MEN1 (0.80) ALDH1A1HPGDMEN1KMT2ASMN1; SMN2
SCHEMBL4471882 0.61 MELK (0.49) ALDH1A1MAPTPOLBLMNAMELK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7585859-B2 PDE4B inhibitors and uses therefor PLEXXIKON, INC. (US) 2009-09-08 US disclosed
US-7585859-B2 PDE4B inhibitors and uses therefor PLEXXIKON, INC. (US) 2009-09-08 US disclosed