SCHEMBL13712759

SCHEMBL13712759

CCN(CC)C(=O)c1ccc2c(c1)Oc1c(OC)cccc1C2=C1CC2CCC(C1)N2C

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 7/20 0.49
OPRD1 P41143 7/20 0.49
CYP1A2 P05177 2/20 0.40
HSP90AA1 P07900 1/20 0.40
HSP90AB1 P08238 1/20 0.40
BLM P54132 1/20 0.40
CYP3A4 P08684 1/20 0.38
NPC1 O15118 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
ALOX15 P16050 1/20 0.37
RAB9A P51151 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4517317 0.89 OPRM1 (0.39) OPRM1OPRD1CYP1A2HSP90AA1HSP90AB1
SCHEMBL490453 0.87 OPRD1 (0.44) OPRM1OPRD1CYP1A2HSP90AA1HSP90AB1
SCHEMBL490111 0.85 OPRD1 (0.53) OPRM1OPRD1
SCHEMBL5096902 0.83 OPRD1 (0.48) OPRM1OPRD1CYP1A2HSP90AA1HSP90AB1
SCHEMBL489911 0.78 OPRM1 (0.48) OPRM1OPRD1
SCHEMBL3177080 0.77 OPRM1 (0.45) OPRM1OPRD1CYP1A2HSP90AA1HSP90AB1
SCHEMBL490182 0.76 OPRD1 (0.40) OPRM1OPRD1
SCHEMBL489974 0.76 OPRD1 (0.45) OPRM1OPRD1HSP90AA1HSP90AB1HPGD
SCHEMBL13627455 0.75 RECQL (0.33) NPC1ALDH1A1HPGDRAB9AHSD17B10
SCHEMBL4509385 0.75 OPRD1 (0.48) OPRM1OPRD1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7589104-B2 Tricyclic-bridged piperidinyline derivatives as §-opioid modulators JANSSEN PHARMACEUTICA NV (BE) 2009-09-15 US disclosed