SCHEMBL1372243

SCHEMBL1372243

Cc1c(C)c2c(C)c3ccoc3cc2oc1=O.NP(O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 4/20 0.43
CYP3A4 P08684 3/20 0.43
ADORA3 P0DMS8 3/20 0.43
CYP1A1 P04798 2/20 0.43
THRB P10828 2/20 0.43
MAPK1 P28482 2/20 0.43
HSD17B3 P37058 3/20 0.42
ALDH1A1 P00352 4/20 0.40
CYP2A6 P11509 2/20 0.40
MAPT P10636 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ALDH2 P05091 2/20 0.39
KDM4E B2RXH2 4/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
HSD17B10 Q99714 2/20 0.38
PGR P06401 1/20 0.38
CYP2D6 P10635 1/20 0.38
KCNA2 P16389 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1002679 0.91 CYP3A4 (0.49) HPGDCYP3A4ADORA3CYP1A1THRB
Hydrochloric Acid SCHEMBL9098003 0.90 ADORA3 (0.48) HPGDCYP3A4ADORA3CYP1A1THRB
SCHEMBL6554781 0.77 SRC (0.45) HPGDCYP3A4ADORA3CYP1A1THRB
SCHEMBL25393535 0.70 ALDH2 (0.50) HPGDCYP3A4ADORA3CYP1A1THRB
SCHEMBL30054772 0.70 ALDH2 (0.50) HPGDCYP3A4ADORA3CYP1A1THRB
SCHEMBL6802035 0.67 ALDH1A1 (0.70) HPGDCYP3A4ADORA3CYP1A1THRB
SCHEMBL698745 0.66 ALDH2 (0.45) HPGDTHRBMAPK1HSD17B3ALDH1A1
SCHEMBL6994969 0.66 ALDH2 (0.56) HPGDCYP3A4ADORA3CYP1A1HSD17B3
SCHEMBL27907872 0.66 ALDH2 (0.47) HPGDCYP3A4MAPK1HSD17B3ALDH1A1
SCHEMBL17525029 0.65 ALDH2 (0.59) HPGDADORA3THRBMAPK1HSD17B3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8658780-B2 Triggered covalent probes for imaging and silencing genetic expression CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2014-02-25 US disclosed
US-20110288148-A1 TRIGGERED COVALENT PROBES FOR IMAGING AND SILENCING GENETIC EXPRESSION NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2011-11-24 US disclosed
US-20100021904-A1 SHIELDED CROSS-LINKING PROBES NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2010-01-28 US disclosed