SCHEMBL13722650

SCHEMBL13722650

C/N=C1/NC(C)(CC(C)C)C(=O)N1CCC1CCN(C(=O)OCc2ccccc2)CC1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
GRIN2B Q13224 10/20 0.42
CYP2D6 P10635 4/20 0.42
CYP2C9 P11712 4/20 0.42
CYP2C19 P33261 1/20 0.42
HTT P42858 1/20 0.41
CYP3A4 P08684 3/20 0.41
FAAH O00519 1/20 0.41
KMT2A Q03164 1/20 0.39
TRPC3 Q13507 2/20 0.39
TRPC7 Q9HCX4 2/20 0.39
XIAP P98170 1/20 0.38
BIRC2 Q13490 1/20 0.38
ENPP2 Q13822 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7512393 0.88 SMN1; SMN2 (0.44) SMN1; SMN2NPC1RAB9AGRIN2BCYP2D6
SCHEMBL13723607 0.82 SMN1; SMN2 (0.35) SMN1; SMN2KMT2A
SCHEMBL7512408 0.81 SMN1; SMN2 (0.46) SMN1; SMN2NPC1RAB9AGRIN2BCYP2D6
SCHEMBL7520459 0.75 KMT2A (0.46) SMN1; SMN2FAAHKMT2A
SCHEMBL17551463 0.74 ACHE (0.36) SMN1; SMN2KMT2A
SCHEMBL7527245 0.72 CHRM4 (0.41) KMT2A
SCHEMBL7528142 0.71 ADAMTS5 (0.40) SMN1; SMN2RAB9ACYP2C9CYP2C19HTT
SCHEMBL13197107 0.71 SMN1; SMN2 (0.65) SMN1; SMN2NPC1RAB9AGRIN2BCYP2D6
SCHEMBL13538207 0.71 SMN1; SMN2 (0.58) SMN1; SMN2NPC1RAB9AGRIN2BCYP2D6
SCHEMBL15140566 0.71 SMN1; SMN2 (0.72) SMN1; SMN2NPC1RAB9AGRIN2BCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1838304-B1 HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS SCHERING CORP (US) 2009-08-19 EP disclosed