SCHEMBL13729992

SCHEMBL13729992

Cc1cc(C#N)c[nH]c1=O

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DPYD Q12882 1/20 0.39
MCL1 Q07820 6/20 0.39
ATAD2 Q6PL18 1/20 0.39
KDM4E B2RXH2 3/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
DAO P14920 4/20 0.37
UPP1 Q16831 1/20 0.35
RECQL P46063 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
PIK3CD O00329 1/20 0.35
PIK3CA P42336 1/20 0.35
PIK3CB P42338 1/20 0.35
GAA P10253 1/20 0.34
BRD4 O60885 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21333260 0.77 MCL1 (0.55) DPYDMCL1KDM4EALDH1A1HPGD
SCHEMBL31399395 0.75 ALDH1A1 (0.44) DPYDMCL1KDM4EALDH1A1HPGD
SCHEMBL1779488 0.75
SCHEMBL29956876 0.75 ENPP2 (0.35) DPYDMCL1KDM4EALDH1A1HPGD
SCHEMBL15358113 0.71 ALDH1A1 (0.44) MCL1KDM4EALDH1A1HPGDDAO
SCHEMBL16649897 0.70 TTR (0.41) KDM4EALDH1A1UPP1RECQLTDP1
SCHEMBL8138214 0.67
SCHEMBL16877088 0.67
SCHEMBL12944279 0.67
SCHEMBL21026422 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015161014-A1 HETEROCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2015-10-22 WO disclosed
EP-2704712-A1 ISOXAZOLINES AS THERAPEUTIC AGENTS AbbVie Inc. (US) 2014-03-12 EP disclosed
WO-2012151158-A1 ISOXAZOLINES AS THERAPEUTIC AGENTS ABBOTT LABORATORIES (US) 2012-11-08 WO disclosed