SCHEMBL13733242

SCHEMBL13733242

FC(F)(F)c1cccc(-c2ccn(Cl)n2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.52
KDM4E B2RXH2 2/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
GABRA1 P14867 1/20 0.52
HPGD P15428 1/20 0.52
GABRG2 P18507 1/20 0.52
GABRB3 P28472 1/20 0.52
GABRA5 P31644 1/20 0.52
GABRA3 P34903 1/20 0.52
GABRA2 P47869 1/20 0.52
HSD17B10 Q99714 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
LMNA P02545 2/20 0.51
IDO1 P14902 1/20 0.50
CTSS P25774 1/20 0.48
CCNA2 P20248 1/20 0.45
CDK2 P24941 1/20 0.45
CDK5 Q00535 1/20 0.45
DYRK1A Q13627 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9383785 0.83 KDM4E (0.56) ALDH1A1KDM4ECYP1A2CYP3A4GABRA1
SCHEMBL26253632 0.80 KDM4E (0.52) ALDH1A1KDM4ECYP1A2CYP3A4GABRA1
SCHEMBL12777946 0.78 ALDH1A1 (0.51) ALDH1A1KDM4ECYP1A2CYP3A4GABRA1
SCHEMBL6697417 0.78 ALDH1A1 (0.66) ALDH1A1KDM4ECYP1A2CYP3A4GABRA1
Benzene SCHEMBL27781609 0.75 KMT2A (0.47) ALDH1A1KMO
SCHEMBL28825532 0.74 CYP1A2 (0.49) ALDH1A1KDM4ECYP1A2CYP3A4GABRA1
SCHEMBL13733343 0.73 KCNH2 (0.39) KDM1A
SCHEMBL29678302 0.73 TSHR (0.58) ALDH1A1IDO1CTSSKDM1AMAOB
SCHEMBL1263144 0.73 TSHR (0.58) ALDH1A1IDO1CTSSKDM1AMAOB
SCHEMBL10850137 0.73 KDR (0.59) ALDH1A1KDM4ECYP1A2CYP3A4GABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2699579-A1 PYRAZOLO [4, 3-D]PYRIMIDINES USEFUL AS KINASE INHIBITORS Origenis GmbH (DE) 2014-02-26 EP claimed
WO-2012143144-A1 PYRAZOLO [4, 3-D] PYRIMIDINES USEFUL AS KINASE INHIBITORS ORIGENIS GMBH (DE) 2012-10-26 WO claimed